RSV ANTIVIRAL PYRAZOLO- AND TRIAZOLO-PYRIMIDINE COMPOUNDS
The invention concerns novel substituted pyrazolo- and triazolo-pyrimidine compounds of formula (I) having antiviral activity, in particular, having an inhibitory activity on the replication of the respiratory syncytial virus (RSV). The invention further concerns pharmaceutical compositions comprisi...
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| Main Authors | , , , , , , , , |
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| Format | Patent |
| Language | English French |
| Published |
19.09.2023
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| Subjects | |
| Online Access | Get full text |
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| Abstract | The invention concerns novel substituted pyrazolo- and triazolo-pyrimidine compounds of formula (I) having antiviral activity, in particular, having an inhibitory activity on the replication of the respiratory syncytial virus (RSV). The invention further concerns pharmaceutical compositions comprising these compounds and the compounds for use in the treatment of respiratory syncytial virus infection.
La présente invention concerne de nouveaux composés de pyrazolo- et triazolo-pyrimidine substitués de formule (I) présentant une activité antivirale, en particulier une activité inhibitrice sur la réplication du virus respiratoire syncytial (VRS). L'invention concerne également des compositions pharmaceutiques comprenant de tels composés, ainsi que lesdits composés destinés à être utilisés dans le traitement d'une infection par le virus respiratoire syncytial. |
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| AbstractList | The invention concerns novel substituted pyrazolo- and triazolo-pyrimidine compounds of formula (I) having antiviral activity, in particular, having an inhibitory activity on the replication of the respiratory syncytial virus (RSV). The invention further concerns pharmaceutical compositions comprising these compounds and the compounds for use in the treatment of respiratory syncytial virus infection.
La présente invention concerne de nouveaux composés de pyrazolo- et triazolo-pyrimidine substitués de formule (I) présentant une activité antivirale, en particulier une activité inhibitrice sur la réplication du virus respiratoire syncytial (VRS). L'invention concerne également des compositions pharmaceutiques comprenant de tels composés, ainsi que lesdits composés destinés à être utilisés dans le traitement d'une infection par le virus respiratoire syncytial. |
| Author | MICHAUT, ANTOINE BENJAMIN LARDEAU, DELPHINE YVONNE RAYMONDE GUILLEMONT, JEROME EMILE GEORGES ROGOVOY, BORIS LANCOIS, DAVID FRANCIS ALAIN ROYMANS, DIRK ANDRE EMMY KOUL, ANIL BICHKO, VADIM RABOISSON, PIERRE JEAN-MARIE BERNARD |
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| DocumentTitleAlternate | COMPOSES DE PYRAZOLO- ET TRIAZOLO-PYRIMIDINE ANTIVIRAUX DU VIRUS RESPIRATOIRE SYNCYTIAL (VRS) |
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| Snippet | The invention concerns novel substituted pyrazolo- and triazolo-pyrimidine compounds of formula (I) having antiviral activity, in particular, having an... |
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| Title | RSV ANTIVIRAL PYRAZOLO- AND TRIAZOLO-PYRIMIDINE COMPOUNDS |
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