NOVEL DICARBOXYLIC ACID DERIVATIVES AS S1P1 RECEPTOR AGONISTS

The present invention relates to new compounds of formula (I) possessing agonistic activity at sphingosine-1 -phosphate (S1 P) receptors, their process of preparation and their use as immunosuppressive agents. The invention is also directed to pharmaceutical compositions containing these compounds a...

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Main Authors ROBERT, PHILIPPE, LECOMTE, JEANNE-MARIE, JIVANI, JIGNESH KANTILAL, CAPET, MARC, PILLAI, MUTHUKUMARAN NATARAJAN, PANCHAL, BHAVESH MOHANBHAI, LEVOIN, NICOLAS, SAMANTA, BISWAJIT, BERREBI-BERTRAND, ISABELLE, ARADHYE, JAYRAJ DILIPBHAI, PAL, RANJAN KUMAR, THENNATI, RAJAMANNAR, SCHWARTZ, JEANARLES
Format Patent
LanguageEnglish
French
Published 18.12.2008
Subjects
CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
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Abstract The present invention relates to new compounds of formula (I) possessing agonistic activity at sphingosine-1 -phosphate (S1 P) receptors, their process of preparation and their use as immunosuppressive agents. The invention is also directed to pharmaceutical compositions containing these compounds and use of these compounds for treatment/prevention of immune medi-ated diseases and conditions or inflammatory diseases and conditions.
AbstractList The present invention relates to new compounds of formula (I) possessing agonistic activity at sphingosine-1 -phosphate (S1 P) receptors, their process of preparation and their use as immunosuppressive agents. The invention is also directed to pharmaceutical compositions containing these compounds and use of these compounds for treatment/prevention of immune medi-ated diseases and conditions or inflammatory diseases and conditions.
Author SCHWARTZ, JEANARLES
CAPET, MARC
LEVOIN, NICOLAS
ROBERT, PHILIPPE
PAL, RANJAN KUMAR
BERREBI-BERTRAND, ISABELLE
JIVANI, JIGNESH KANTILAL
LECOMTE, JEANNE-MARIE
SAMANTA, BISWAJIT
PILLAI, MUTHUKUMARAN NATARAJAN
THENNATI, RAJAMANNAR
ARADHYE, JAYRAJ DILIPBHAI
PANCHAL, BHAVESH MOHANBHAI
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– fullname: PAL, RANJAN KUMAR
– fullname: THENNATI, RAJAMANNAR
– fullname: SCHWARTZ, JEANARLES
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DocumentTitleAlternate NOUVEAUX DERIVES D'ACIDE DICARBOXYLIQUE UTILISES COMME AGONISTES DU RECEPTEUR S1P1
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Snippet The present invention relates to new compounds of formula (I) possessing agonistic activity at sphingosine-1 -phosphate (S1 P) receptors, their process of...
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HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
Title NOVEL DICARBOXYLIC ACID DERIVATIVES AS S1P1 RECEPTOR AGONISTS
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