BENZYLTHIAZOLONE INHIBITORS OF ESTROGEN-RELATED RECEPTORS (ERR)

Compounds for use in compositions and methods for modulating the activity of nuclear receptors are provided. In particular, compounds for use in compositions and methods for modulating the estrogen related receptors are provided. In one embodiment, the compounds provided herein are ERR modulators. I...

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Bibliographic Details
Main Authors MOHAN, RAJU, MARTIN, RICHARD, STEVENS, WILLIAM C., JR, BUSCH, BRETT B, NYMAN, MICHAEL CHARLES
Format Patent
LanguageEnglish
French
Published 20.05.2014
Subjects
CHEMISTRY
HETEROCYCLIC COMPOUNDS
METALLURGY
ORGANIC CHEMISTRY
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Summary:Compounds for use in compositions and methods for modulating the activity of nuclear receptors are provided. In particular, compounds for use in compositions and methods for modulating the estrogen related receptors are provided. In one embodiment, the compounds provided herein are ERR modulators. In another embodiment, the compounds provided herein are agonists, partial agonists, antagonists. or inverse agonists of ERR or ERR. In certain embodiments, the compounds of the invention, as described above in the Summary of the Invention, are compounds of formula (I).
Bibliography:Application Number: CA20052583271