DIHYDROPYRIMIDINES

The invention relates to compounds of general formula (I) or general formula (Ia). The invention also relates to methods for producing said compounds of general formula (I) or (Ia) and to their use as medicaments, especially for treating and preventing hepatitis B. The compounds of the formula (I) o...

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Main Authors WEBER, OLAF, DERES, KARL, PAESSENS, ARNOLD, LOTTMANN, STEFAN, KRAMER, THOMAS, GRAEF, ERWIN, NIEWOHNER, ULRICH, STOLTEFUSS, JURGEN, STOLTING, JORN, GOLDMANN, SIEGFRIED, SCHLEMMER, KARL-HEINZ
Format Patent
LanguageEnglish
French
Published 23.09.2008
Subjects
CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
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Summary:The invention relates to compounds of general formula (I) or general formula (Ia). The invention also relates to methods for producing said compounds of general formula (I) or (Ia) and to their use as medicaments, especially for treating and preventing hepatitis B. The compounds of the formula (I) or (Ia) have the structure: (see formula I, II ) or a salt thereof, wherein R1 is a cyclic moiety; R2 is hydrogen, -OH, C1-C6 alkoxycarbonyl, etc.; R3 is hydrogen, amino, etc.; R4 is hydrogen, alkyl, alkenyl, etc.; and R5 is substituted pyridyl.
Bibliography:Application Number: CA19992328780