1,5-BENZODIAZEPINE DERIVATIVES

1,5-Benzodiazepine derivatives represented by formula (I), salts thereof, and medicines containing the same as the active ingredient: (see formula I) [wherein R1 represents a hydrogen atom, a lower alkyl group, a lower alkoxyl group, or a halogen atom; each of R2 and R3, which may be the same or dif...

Full description

Saved in:
Bibliographic Details
Main Authors SHINOZAKI, KATSUO, MIURA, NAOYOSHI, MAEDA, KIYOTO, YONETA, TOMOYUKI, MURATA, MASAKAZU
Format Patent
LanguageEnglish
French
Published 14.11.2006
Subjects
CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
Online AccessGet full text

Cover

More Information
Summary:1,5-Benzodiazepine derivatives represented by formula (I), salts thereof, and medicines containing the same as the active ingredient: (see formula I) [wherein R1 represents a hydrogen atom, a lower alkyl group, a lower alkoxyl group, or a halogen atom; each of R2 and R3, which may be the same or different, represents a hydrogen atom, an alkenyl group, an alkyl group, a phenyl group, an acyl group, etc; and each of R4 and R5, which may be the same or different, represents a hydrogen atom, an alkyl group, a carboxyl group, etc.]. The compounds exhibit excellent gastrin and/or CCK-B receptor antagonism and are useful as remedies for gastric ulcer and gastrointestinal movement disorder.
Bibliography:Application Number: CA19972274669