Benzimidazole derivatives

According to a first aspect of the invention there is provided compounds of formula (I):wherein:R1 is hydroxy; O-acetyl; or a halo atom;R2 is hydroxy; O-acetyl; or a halo atom;R3 is hydrogen; a halo atom; azido; C2-6alkenyl; C2-6alkynyl; C6-14aryl C2-6alkenyl; C6-14arylC2-6alkynyl -NR8R9 (where R8 a...

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Bibliographic Details
Main Authors JOSEPH HOWING CHAN, LEROY B TOWNSEND, GEORGE ANDREW FREEMAN, GEORGE WALTER KOSZALKA, STANLEY DAWES CHAMBERLAIN, JOHN C DRACH, JEFFREY H. TIDWELL
Format Patent
LanguageEnglish
Published 08.09.1998
Edition6
Subjects
CHEMISTRY
DERIVATIVES THEREOF
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
NUCLEIC ACIDS
NUCLEOSIDES
NUCLEOTIDES
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
SUGARS
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Summary:According to a first aspect of the invention there is provided compounds of formula (I):wherein:R1 is hydroxy; O-acetyl; or a halo atom;R2 is hydroxy; O-acetyl; or a halo atom;R3 is hydrogen; a halo atom; azido; C2-6alkenyl; C2-6alkynyl; C6-14aryl C2-6alkenyl; C6-14arylC2-6alkynyl -NR8R9 (where R8 and R9 may be the same or different and are hydrogen, C1-8alkyl, cyanoC1-8alkyl, hydroxyC1-8alkyl, haloC1-8alkyl, C3-7cycloalkyl, C1-8alkylC3-7cycloalkyl, C2-6alkenyl, C3-7cycloalkylC1-8alkyl, C2-6alkynyl, C6-14aryl, C6-14arylC1-8alkyl, heterocycleC1-8alkyl, C1-8alkylcarbonyl, C6-14arylsulfonyl, C1-8alkysulfonyl, or R8R9 together with the N atom to which they are attached form a 3,4,5 or 6 membered heterocyclic ring); -OR10 (where R10 is hydrogen, C1-8alkyl, C6-14aryl, or C6-14arylC1-8alkyl, C2-6alkenyl, C2-6alkynyl, C6-14aryl C2-6alkenyl or C6-14arylC2-6alkynyl); or -SR11 (where R11 is hydrogen, C1-8alkyl, C6-14aryl, or C6-14arylC1-8alkyl).
Bibliography:Application Number: AU19980000622