Non-steroidal estrogen receptor ligands

Novel non-steroidal estrogen receptor ligands and methods of synthesis are disclosed. The novel molecules are intended for use in therapeutic preparations for the treatment of estrogen receptor related disease states. The compounds specified are tetra-cyclic derivatives and have been shown to be ant...

Full description

Saved in:
Bibliographic Details
Main Authors JEFFRY LAWRENCE LOWELL, JOHN WHELAN, STEFAN KWIATKOWSKI, JULIE MERCURE, NATALIE LAZAROWYCH, KRZYSZTOF PUPEK, JONATHAN MARTIN SCHMIDT, SHUGUANG ZHU
Format Patent
LanguageEnglish
Published 04.09.2002
Edition7
Subjects
CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
Online AccessGet full text

Cover

Abstract Novel non-steroidal estrogen receptor ligands and methods of synthesis are disclosed. The novel molecules are intended for use in therapeutic preparations for the treatment of estrogen receptor related disease states. The compounds specified are tetra-cyclic derivatives and have been shown to be antiproliferative against human estrogen-dependent cancer cells and to have good binding affinity for the estrogen receptor.
AbstractList Novel non-steroidal estrogen receptor ligands and methods of synthesis are disclosed. The novel molecules are intended for use in therapeutic preparations for the treatment of estrogen receptor related disease states. The compounds specified are tetra-cyclic derivatives and have been shown to be antiproliferative against human estrogen-dependent cancer cells and to have good binding affinity for the estrogen receptor.
Author SHUGUANG ZHU
JEFFRY LAWRENCE LOWELL
KRZYSZTOF PUPEK
STEFAN KWIATKOWSKI
NATALIE LAZAROWYCH
JULIE MERCURE
JONATHAN MARTIN SCHMIDT
JOHN WHELAN
Author_xml – fullname: JEFFRY LAWRENCE LOWELL
– fullname: JOHN WHELAN
– fullname: STEFAN KWIATKOWSKI
– fullname: JULIE MERCURE
– fullname: NATALIE LAZAROWYCH
– fullname: KRZYSZTOF PUPEK
– fullname: JONATHAN MARTIN SCHMIDT
– fullname: SHUGUANG ZHU
BookMark eNrjYmDJy89L5WRQ98vP0y0uSS3Kz0xJzFFILS4pyk9PzVMoSk1OLSjJL1LIyUxPzEsp5mFgTUvMKU7lhdLcDMpuriHOHrqpBfnxqcUFicmpeakl8Y6hRgYGRkbGFsaGJo6GxsSpAgBKrSq6
ContentType Patent
DBID EVB
DatabaseName esp@cenet
DatabaseTitleList
Database_xml – sequence: 1
  dbid: EVB
  name: esp@cenet
  url: http://worldwide.espacenet.com/singleLineSearch?locale=en_EP
  sourceTypes: Open Access Repository
DeliveryMethod fulltext_linktorsrc
Discipline Medicine
Chemistry
Sciences
Edition 7
ExternalDocumentID AU2002238314A1
GroupedDBID EVB
ID FETCH-epo_espacenet_AU2002238314A13
IEDL.DBID EVB
IngestDate Fri Jul 19 15:05:20 EDT 2024
IsOpenAccess true
IsPeerReviewed false
IsScholarly false
Language English
LinkModel DirectLink
MergedId FETCHMERGED-epo_espacenet_AU2002238314A13
Notes Application Number: AU20020238314
OpenAccessLink https://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20020904&DB=EPODOC&CC=AU&NR=2002238314A1
ParticipantIDs epo_espacenet_AU2002238314A1
PublicationCentury 2000
PublicationDate 20020904
PublicationDateYYYYMMDD 2002-09-04
PublicationDate_xml – month: 09
  year: 2002
  text: 20020904
  day: 04
PublicationDecade 2000
PublicationYear 2002
RelatedCompanies NANODESIGN INC
RelatedCompanies_xml – name: NANODESIGN INC
Score 2.5582142
Snippet Novel non-steroidal estrogen receptor ligands and methods of synthesis are disclosed. The novel molecules are intended for use in therapeutic preparations for...
SourceID epo
SourceType Open Access Repository
SubjectTerms CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
Title Non-steroidal estrogen receptor ligands
URI https://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20020904&DB=EPODOC&locale=&CC=AU&NR=2002238314A1
hasFullText 1
inHoldings 1
isFullTextHit
isPrint
link http://utb.summon.serialssolutions.com/2.0.0/link/0/eLvHCXMwfV1LS8NAEB5KFfWmVfFRJaDEU7BJNhtzKNLmQRFMi7TSW9lkdyUQktBG_PtOlkZ76m2ZhX0yj29nZwbgMZGuxaklDcodYRBic8OjL9xITSZTtJAF0pvfFjGdLMjb0ll2IG9jYVSe0B-VHBE5KkV-r5W8rv4fsQL1t3LznGRIKl-j-TDQW3RsDTy89GA8DGfTYOrrvo9IUo8_VB9qJ9skI8RKB2hIuw0_hJ_jJi6l2lUq0SkcznC8oj6Djih6cOy3tdd6cPS-dXljc8t9m3N4isvCaBIblBlnuYbyfF3i_WsotESF2FnLs68mcvcCHqJw7k8MnHH1t8HVaLG7PPsSugj9xRVozCWMuFQyiznEHNiJJK5FpccEN1OEkNfQ3zfSzf7uWzhRtU2Ue6QP3Xr9Le5QxdbJvTqZX_h4fuE
link.rule.ids 230,309,783,888,25576,76876
linkProvider European Patent Office
linkToHtml http://utb.summon.serialssolutions.com/2.0.0/link/0/eLvHCXMwfV1LT4NAEJ401VhvWjVWq5Jo8EQssIAcGtPyCGpLG0NNb80CiyEhQFqMf99hU7Sn3jazyT4zj29nZwbgIUwMJdaVRNJjjUmEqLFk6s-xFMk0idBCZkivf1v4urcgb0tt2YKsiYXheUJ_eHJE5KgI-b3i8rr8f8Sy-d_KzVOYIql4cYOhLTboWBmYeOn2eOjMZ_bMEi0LkaTof_A-1E6qTEaIlQ7QyDZqfnA-x3VcSrmrVNwTOJzjeHl1Ci2Wd6FjNbXXunA03bq8sbnlvs0ZPPpFLtWJDYo0ppmA8nxd4P0LKLRYidhZyNKvOnL3HO5dJ7A8CWdc_W1wNVrsLk-9gDZCf3YJAjUIJYaeUIVqRB6oYUIMRU9MymI5QgjZg_6-ka72d99Bxwumk9Xk1X-_hmNe54S7SvrQrtbf7AbVbRXe8lP6BRbZgdQ
openUrl ctx_ver=Z39.88-2004&ctx_enc=info%3Aofi%2Fenc%3AUTF-8&rfr_id=info%3Asid%2Fsummon.serialssolutions.com&rft_val_fmt=info%3Aofi%2Ffmt%3Akev%3Amtx%3Apatent&rft.title=Non-steroidal+estrogen+receptor+ligands&rft.inventor=JEFFRY+LAWRENCE+LOWELL&rft.inventor=JOHN+WHELAN&rft.inventor=STEFAN+KWIATKOWSKI&rft.inventor=JULIE+MERCURE&rft.inventor=NATALIE+LAZAROWYCH&rft.inventor=KRZYSZTOF+PUPEK&rft.inventor=JONATHAN+MARTIN+SCHMIDT&rft.inventor=SHUGUANG+ZHU&rft.date=2002-09-04&rft.externalDBID=A1&rft.externalDocID=AU2002238314A1