VERFAHREN ZUR HERSTELLUNG VON CHINAZOLINDERIVATEN

Procedure for preparation of quinazoline derivatives. The invention is related to a procedure for the preparation of quinazoline derivatives of general formula i, in which rbs1 and rbs2 can be equal or different and represent hydrogen or lower rent, or jointly form a group ethylene or trimethylene,...

Full description

Saved in:
Bibliographic Details
Main Authors SZTUHAR ILONA DR, FEKETE MARTON DR, PONGO LASZLO . DR, REITER JOZSEF DR, CSOERGO MARGIT DR, GOERGENYI FRIGYES DR
Format Patent
LanguageGerman
Published 26.09.1994
Edition5
Subjects
CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOIDCHEMISTRY
CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PERFORMING OPERATIONS
PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
THEIR RELEVANT APPARATUS
TRANSPORTING
Online AccessGet full text

Cover

More Information
Summary:Procedure for preparation of quinazoline derivatives. The invention is related to a procedure for the preparation of quinazoline derivatives of general formula i, in which rbs1 and rbs2 can be equal or different and represent hydrogen or lower rent, or jointly form a group ethylene or trimethylene, yn is 2 or 3, characterized by the reaction of a 1,2 dimetoxy phenyl 4 istitiourea derivative, with a diamincarboxifuran derivative, eventually substituted, and posterior cyclation, thermal or catalytic, of the compound so obtained. The invention is also related, with the preparation of the intermediate reaction compounds. The compounds object of this invention have interesting properties pharmaceutical as antihypertensive and blockers of si1 receptors. (Machine-translation by Google Translate, not legally binding)
Bibliography:Application Number: AT93190