4-(( R )-2-{[6-(( S )-3-Methoxypyrrolidin-1-yl)-2-phenylpyrimidine-4-carbonyl]amino}-3-phosphonopropionyl)piperazine-1-carboxylic Acid Butyl Ester (ACT-246475) and Its Prodrug (ACT-281959), a Novel P2Y 12 Receptor Antagonist with a Wider Therapeutic Window in the Rat Than Clopidogrel
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Published in | Journal of medicinal chemistry Vol. 58; no. 23; pp. 9133 - 9153 |
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Main Authors | , , , , , , , , , , |
Format | Journal Article |
Language | English |
Published |
10.12.2015
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Online Access | Get full text |
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ISSN: | 0022-2623 1520-4804 |
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DOI: | 10.1021/acs.jmedchem.5b00933 |