4-(( R )-2-{[6-(( S )-3-Methoxypyrrolidin-1-yl)-2-phenylpyrimidine-4-carbonyl]amino}-3-phosphonopropionyl)piperazine-1-carboxylic Acid Butyl Ester (ACT-246475) and Its Prodrug (ACT-281959), a Novel P2Y 12 Receptor Antagonist with a Wider Therapeutic Window in the Rat Than Clopidogrel

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Bibliographic Details
Published inJournal of medicinal chemistry Vol. 58; no. 23; pp. 9133 - 9153
Main Authors Caroff, Eva, Hubler, Francis, Meyer, Emmanuel, Renneberg, Dorte, Gnerre, Carmela, Treiber, Alexander, Rey, Markus, Hess, Patrick, Steiner, Beat, Hilpert, Kurt, Riederer, Markus A.
Format Journal Article
LanguageEnglish
Published 10.12.2015
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ISSN:0022-2623
1520-4804
DOI:10.1021/acs.jmedchem.5b00933