Multiparameter Optimization in CNS Drug Discovery: Design of Pyrimido[4,5- d ]azepines as Potent 5-Hydroxytryptamine 2C (5-HT 2C ) Receptor Agonists with Exquisite Functional Selectivity over 5-HT 2A and 5-HT 2B Receptors

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Bibliographic Details
Published inJournal of medicinal chemistry Vol. 57; no. 12; pp. 5258 - 5269
Main Authors Storer, R. Ian, Brennan, Paul E., Brown, Alan D., Bungay, Peter J., Conlon, Kelly M., Corbett, Matthew S., DePianta, Robert P., Fish, Paul V., Heifetz, Alexander, Ho, Danny K. H., Jessiman, Alan S., McMurray, Gordon, de Oliveira, Cesar Augusto F., Roberts, Lee R., Root, James A., Shanmugasundaram, Veerabahu, Shapiro, Michael J., Skerten, Melanie, Westbrook, Dominique, Wheeler, Simon, Whitlock, Gavin A., Wright, John
Format Journal Article
LanguageEnglish
Published 26.06.2014
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ISSN:0022-2623
1520-4804
DOI:10.1021/jm5003292