黄柏水提物联合抗菌药对产ESBLs大肠杆菌的抑菌效果
【目的】探讨黄柏水提物与抗菌药联用对产超广谱β-内酰胺酶(ESBLs)大肠杆菌的抑制效果,为黄柏的综合开发利用提供参考依据。【方法】采用二倍微量肉汤稀释法测定黄柏水提物与抗菌药的最小抑菌浓度(MIC),并采用微量棋盘稀释法测定黄柏水提物与抗菌药联用后的分级抑菌浓度指数(FICI)。【结果】黄柏水提物对产ESBLs大肠杆菌的MIC为500 mg/m L,黄柏水提物与头孢曲松钠、阿莫西林、痢菌净、磺胺间甲氧嘧啶、头孢噻呋钠、头孢他啶、氟苯尼考、环丙沙星、诺氟沙星、左旋氧氟沙星、克林沙星、加替沙星、头孢噻肟联用后的FICI为0.50~2.01,其中,黄柏水提物与阿莫西林、头孢曲松钠、头孢噻呋钠、头孢...
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Published in | 南方农业学报 Vol. 47; no. 3; pp. 500 - 505 |
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Main Author | |
Format | Journal Article |
Language | Chinese |
Published |
广西大学 动物科学技术学院,南宁,530005
2016
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Subjects | |
Online Access | Get full text |
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Abstract | 【目的】探讨黄柏水提物与抗菌药联用对产超广谱β-内酰胺酶(ESBLs)大肠杆菌的抑制效果,为黄柏的综合开发利用提供参考依据。【方法】采用二倍微量肉汤稀释法测定黄柏水提物与抗菌药的最小抑菌浓度(MIC),并采用微量棋盘稀释法测定黄柏水提物与抗菌药联用后的分级抑菌浓度指数(FICI)。【结果】黄柏水提物对产ESBLs大肠杆菌的MIC为500 mg/m L,黄柏水提物与头孢曲松钠、阿莫西林、痢菌净、磺胺间甲氧嘧啶、头孢噻呋钠、头孢他啶、氟苯尼考、环丙沙星、诺氟沙星、左旋氧氟沙星、克林沙星、加替沙星、头孢噻肟联用后的FICI为0.50~2.01,其中,黄柏水提物与阿莫西林、头孢曲松钠、头孢噻呋钠、头孢他啶、头孢噻肟、痢菌净联用存在相加作用,与氟苯尼考联用存在协同作用,与诺氟沙星、左旋氧氟沙星、克林沙星、磺胺间甲氧嘧啶间为无关作用,与环丙沙星、加替沙星联用呈拮抗作用。【结论】黄柏水提物与青霉素类、第三代头孢菌素、痢菌净、氟苯尼考联用是通过相加或协同作用提高药物对产ESBLs大肠杆菌的抑制效果,但不宜与喹诺酮类抗菌药联合用药。 |
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AbstractList | 【目的】探讨黄柏水提物与抗菌药联用对产超广谱β-内酰胺酶(ESBLs)大肠杆菌的抑制效果,为黄柏的综合开发利用提供参考依据。【方法】采用二倍微量肉汤稀释法测定黄柏水提物与抗菌药的最小抑菌浓度(MIC),并采用微量棋盘稀释法测定黄柏水提物与抗菌药联用后的分级抑菌浓度指数(FICI)。【结果】黄柏水提物对产ESBLs大肠杆菌的MIC为500 mg/m L,黄柏水提物与头孢曲松钠、阿莫西林、痢菌净、磺胺间甲氧嘧啶、头孢噻呋钠、头孢他啶、氟苯尼考、环丙沙星、诺氟沙星、左旋氧氟沙星、克林沙星、加替沙星、头孢噻肟联用后的FICI为0.50~2.01,其中,黄柏水提物与阿莫西林、头孢曲松钠、头孢噻呋钠、头孢他啶、头孢噻肟、痢菌净联用存在相加作用,与氟苯尼考联用存在协同作用,与诺氟沙星、左旋氧氟沙星、克林沙星、磺胺间甲氧嘧啶间为无关作用,与环丙沙星、加替沙星联用呈拮抗作用。【结论】黄柏水提物与青霉素类、第三代头孢菌素、痢菌净、氟苯尼考联用是通过相加或协同作用提高药物对产ESBLs大肠杆菌的抑制效果,但不宜与喹诺酮类抗菌药联合用药。 S853.74; [目的]探讨黄柏水提物与抗菌药联用对产超广谱β-内酰胺酶(ESBLs)大肠杆菌的抑制效果,为黄柏的综合开发利用提供参考依据.[方法]采用二倍微量肉汤稀释法测定黄柏水提物与抗菌药的最小抑菌浓度(MIC),并采用微量棋盘稀释法测定黄柏水提物与抗菌药联用后的分级抑菌浓度指数(FICI).[结果]黄柏水提物对产ESBLs大肠杆菌的MIC为500 mg/mL,黄柏水提物与头孢曲松钠、阿莫西林、痢菌净、磺胺间甲氧嘧啶、头孢噻呋钠、头孢他啶、氟苯尼考、环丙沙星、诺氟沙星、左旋氧氟沙星、克林沙星、加替沙星、头孢噻肟联用后的FICI为0.50~2.01,其中,黄柏水提物与阿莫西林、头孢曲松钠、头孢噻呋钠、头孢他啶、头孢噻肟、痢菌净联用存在相加作用,与氟苯尼考联用存在协同作用,与诺氟沙星、左旋氧氟沙星、克林沙星、磺胺间甲氧嘧啶间为无关作用,与环丙沙星、加替沙星联用呈拮抗作用.[结论]黄柏水提物与青霉素类、第三代头孢菌素、痢菌净、氟苯尼考联用是通过相加或协同作用提高药物对产ESBLs大肠杆菌的抑制效果,但不宜与喹诺酮类抗菌药联合用药. |
Author | 徐素萍 刘增援 吴永继 梁政 潘婕 孙燕杰 宋剑武 黄凯 司红彬 |
AuthorAffiliation | 广西大学动物科学技术学院,南宁530005 |
AuthorAffiliation_xml | – name: 广西大学 动物科学技术学院,南宁,530005 |
Author_xml | – sequence: 1 fullname: 徐素萍 刘增援 吴永继 梁政 潘婕 孙燕杰 宋剑武 黄凯 司红彬 |
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Copyright | Copyright © Wanfang Data Co. Ltd. All Rights Reserved. |
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DOI | 10.3969/j:issn.2095-1191.2016.03.500 |
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DocumentTitleAlternate | Antibacterial effects of Phellodendron amurense Rupr water extracts combined with antimicrobials on ESBLs-producing Escherichia coli |
DocumentTitle_FL | Antibacterial effects of Phellodendron amurense Rupr water extracts combined with antimicrobials on ESBLs-producing Escherichia coli |
EndPage | 505 |
ExternalDocumentID | gxnykx201603031 668535012 |
GrantInformation_xml | – fundername: 国家自然科学基金项目; 国家科技支撑计划项目; 广西自然科学基金项目; 广西科学研究与技术开发计划项目 funderid: (31460675); (2012BAD25B04); (2013GXNSFA-A019070); (0992014-2) |
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Keywords | 联合用药 checkerboard microdilution method drug combination ESBLs-producing Escherichia coli 黄柏 抗菌药 产ESBLs大肠杆菌 FICI Phellodendron amurense Rupr antibacterial 微量棋盘稀释法 fractional inhibitory concentration index (FICI) |
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Notes | Objective】The present experiment was conducted to investigate antibacterial effects of Phellodendron amurense Rupr water extracts combined with antimicrobials on ESBLs-producing Escherichia coli, in order to provide reference for comprehensive exploitation and utilization of P. amurense. 【Method】The minimal inhibitory concentration(MIC)of P. amurense water extracts combined with antibacterial agents were determined by double broth microdilution method.And the fractional inhibitory concentration index(FICI) of P. amurense water extracts combined with antibacterial agents to were determined by checkerboard microdilution method. 【Result】The MIC of P. amurense water extracts was 500 mg/m L.The FICI of P. amurense water extracts combined with ceftriaxone sodium, amoxicillin, mequindox, sulfamonomethoxine,ceftiofur sodium, ceftazidime, florfenicol, ciprofloxacin, norfloxacin, levofloxacin, clinafloxacin, gatifloxacin and cefotaxime ranged from 0.50 to 2.01. There was additive effect between P. amurense water extrac |
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PublicationTitle | 南方农业学报 |
PublicationTitleAlternate | Journal of Southern Agriculture |
PublicationTitle_FL | Journal of Southern Agriculture |
PublicationYear | 2016 |
Publisher | 广西大学 动物科学技术学院,南宁,530005 |
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SubjectTerms | FICI 产ESBLs大肠杆菌 微量棋盘稀释法 抗菌药 联合用药 黄柏 |
Title | 黄柏水提物联合抗菌药对产ESBLs大肠杆菌的抑菌效果 |
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