Palladium-catalyzed synthesis of indoles via intramolecular Heck reaction

Highly effective Pd-catalyzed synthesis of indoles from 2-halo-anilines and allyl bromides via intramolecular Heck reaction in the presence of P(OPh)3 as the ligand is described. [Display omitted] •Synthesis of indoles•Intramolecular Heck reaction•Readily available P(OPh)3 as the ligand•Cyclization...

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Bibliographic Details
Published inCatalysis communications Vol. 38; pp. 21 - 25
Main Authors Yang, Hailong, Sun, Peng, Zhu, Yan, Yan, Hong, Lu, Linhua, Liu, Defu, Rong, Guangwei, Mao, Jincheng
Format Journal Article
LanguageEnglish
Published Elsevier B.V 05.08.2013
Subjects
Allyl bromides
Coupling reactions
Cyclization
Heck reaction
Palladium catalysis
Heck reaction
Coupling reactions
Cyclization
Allyl bromides
Palladium catalysis
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Summary:Highly effective Pd-catalyzed synthesis of indoles from 2-halo-anilines and allyl bromides via intramolecular Heck reaction in the presence of P(OPh)3 as the ligand is described. [Display omitted] •Synthesis of indoles•Intramolecular Heck reaction•Readily available P(OPh)3 as the ligand•Cyclization
ISSN:1566-7367
1873-3905
DOI:10.1016/j.catcom.2013.04.001