In search of potent histamine-3 receptor antagonists

Starting with modafinil, an alertness and wake-promoting agent but inactive in histamine 3 receptor (H3R) binding assay, a series of potent H3 receptor antagonists were developed.

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Bibliographic Details
Published inJournal of King Saud University. Science Vol. 27; no. 2; pp. 189 - 192
Main Author Chatterjee, Sankar
Format Journal Article
LanguageEnglish
Published Elsevier B.V 01.04.2015
Elsevier
Subjects
Antagonist
Histamine-3
Modafinil
Suzuki reaction
Antagonist
Modafinil
Histamine-3
Suzuki reaction
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Summary:Starting with modafinil, an alertness and wake-promoting agent but inactive in histamine 3 receptor (H3R) binding assay, a series of potent H3 receptor antagonists were developed.
ISSN:1018-3647
DOI:10.1016/j.jksus.2014.09.003