Rhodium-Catalyzed Regioselective C–H Chlorination of 7‑Azaindoles Using 1,2-Dichloroethane
An unexpected rhodium-catalyzed regioselective C–H chlorination of 7-azaindoles was developed using 1,2-dichloroethane (DCE) as a chlorinating agent and 7-azaindole as the directing group. This protocol provides an efficient access to ortho-chlorinated azaindoles with operational simplicity, good fu...
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Published in | Organic letters Vol. 16; no. 20; pp. 5294 - 5297 |
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Main Authors | , , , , |
Format | Journal Article |
Language | English |
Published |
WASHINGTON
American Chemical Society
17.10.2014
Amer Chemical Soc |
Subjects | |
Online Access | Get full text |
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