A Remarkably Simple Protocol for the N-Formylation of Amino Acid Esters and Primary Amines

A simple, convenient, and wide scope protocol for the N-formylation of amino acid esters and primary amines has been developed utilizing only imidazole in warm DMF.

Saved in:
Bibliographic Details
Published inOrganic letters Vol. 13; no. 15; pp. 3952 - 3955
Main Authors Suchý, Mojmír, Elmehriki, Adam A. H, Hudson, Robert H. E
Format Journal Article
LanguageEnglish
Published WASHINGTON American Chemical Society 05.08.2011
Amer Chemical Soc
Subjects
Amines - chemistry
Amino Acids - chemistry
Chemistry
Chemistry, Organic
Esters - chemistry
Formates - chemistry
Imidazoles - chemistry
Molecular Structure
Physical Sciences
Science & Technology
FORMIC-ACID
DESIGN
DIMETHYLFORMAMIDE
COMPLEXES
AGENTS
IMIDAZOLE
DERIVATIVES
PEPTIDE
Online AccessGet full text

Cover

More Information
Summary:A simple, convenient, and wide scope protocol for the N-formylation of amino acid esters and primary amines has been developed utilizing only imidazole in warm DMF.
Bibliography:ObjectType-Article-1
SourceType-Scholarly Journals-1
ObjectType-Feature-2
content type line 23
ISSN:1523-7060
1523-7052
DOI:10.1021/ol201475j