Novel heterocyclic-substituted benzofuran histamine H3 receptor antagonists : In vitro properties, drug-likeness, and behavioral activity Art Hancock memorial special issue: Adrenergic and histaminergic pharmacology
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Published in | Biochemical pharmacology Vol. 73; no. 8; pp. 1243 - 1255 |
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Main Authors | , , , , , , , , , , , , , , , , , , , , , , , , |
Format | Journal Article |
Language | English |
Published |
New York, NY
Elsevier Science
2007
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Subjects | |
Online Access | Get full text |
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Author | WETTER, Jill M GFESSER, Gregory A GAGNE, Gerard D MARSH, Kennan C MILICIC, Ivan XIAOQING DENG MILLER, Thomas R DIAZ, Gilbert J WITTE, David G MOLESKY, Angela L BUCKLEY, Michael J DIEHL, Marilyn S LIPING PAN ROBERTS, Ellen M HANCOCK, Arthur A KRUEGER, Kathleen M FOX, Gerard B COWART, Marlon BRIONI, Jorge D BROWMAN, Kaitlin E KOMATER, Victoria A ESBENSHADE, Timothy A FAGHIH, Ramin DELIANG ZHOU BARANOWSKI, John L |
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IL 60064-6123, United States – sequence: 11 givenname: Marilyn S surname: DIEHL fullname: DIEHL, Marilyn S organization: GPRD_AP9a/216, Department of Neuroscience Research, Abbott Laboratories, Abbott Park, IL 60064-6123, United States – sequence: 12 givenname: Jill M surname: WETTER fullname: WETTER, Jill M organization: GPRD_AP9a/216, Department of Neuroscience Research, Abbott Laboratories, Abbott Park, IL 60064-6123, United States – sequence: 13 givenname: Kaitlin E surname: BROWMAN fullname: BROWMAN, Kaitlin E organization: GPRD_AP9a/216, Department of Neuroscience Research, Abbott Laboratories, Abbott Park, IL 60064-6123, United States – sequence: 14 givenname: Kennan C surname: MARSH fullname: MARSH, Kennan C organization: GPRD_AP9a/216, Department of Neuroscience Research, Abbott Laboratories, Abbott Park, IL 60064-6123, United States – sequence: 15 givenname: Gerard B surname: FOX fullname: FOX, Gerard B organization: GPRD_AP9a/216, Department of Neuroscience Research, Abbott Laboratories, Abbott Park, IL 60064-6123, United States – sequence: 16 givenname: Jorge D surname: BRIONI fullname: BRIONI, Jorge D organization: GPRD_AP9a/216, Department of Neuroscience Research, Abbott Laboratories, Abbott Park, IL 60064-6123, United States – sequence: 17 givenname: Timothy A surname: ESBENSHADE fullname: ESBENSHADE, Timothy A organization: GPRD_AP9a/216, Department of Neuroscience Research, Abbott Laboratories, Abbott Park, IL 60064-6123, United States – sequence: 18 givenname: Arthur A surname: HANCOCK fullname: HANCOCK, Arthur A organization: GPRD_AP9a/216, Department of Neuroscience Research, Abbott Laboratories, Abbott Park, IL 60064-6123, United States – sequence: 19 givenname: Ramin surname: FAGHIH fullname: FAGHIH, Ramin organization: GPRD_AP9a/216, Department of Neuroscience Research, Abbott Laboratories, Abbott Park, IL 60064-6123, United States – sequence: 20 givenname: Thomas R surname: MILLER fullname: MILLER, Thomas R organization: GPRD_AP9a/216, Department of Neuroscience Research, Abbott Laboratories, Abbott Park, IL 60064-6123, United States – sequence: 21 givenname: Ivan surname: MILICIC fullname: MILICIC, Ivan organization: GPRD_AP9a/216, Department of Neuroscience Research, Abbott Laboratories, Abbott Park, IL 60064-6123, United States – sequence: 22 givenname: John L surname: BARANOWSKI fullname: BARANOWSKI, John L organization: GPRD_AP9a/216, Department of Neuroscience Research, Abbott Laboratories, Abbott Park, IL 60064-6123, United States – sequence: 23 givenname: Kathleen M surname: KRUEGER fullname: KRUEGER, Kathleen M organization: GPRD_AP9a/216, Department of Neuroscience Research, Abbott Laboratories, Abbott Park, IL 60064-6123, United States – sequence: 24 givenname: David G surname: WITTE fullname: WITTE, David G organization: GPRD_AP9a/216, Department of Neuroscience Research, Abbott Laboratories, Abbott Park, IL 60064-6123, United States – sequence: 25 givenname: Angela L surname: MOLESKY fullname: MOLESKY, 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Keywords | Drug Histamine A-688057 H3 receptor H3 histamine receptor Central nervous system CNS Antagonist Behavior In vitro Biological activity Heterocyclic compound |
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Subtitle | Art Hancock memorial special issue: Adrenergic and histaminergic pharmacology |
Title | Novel heterocyclic-substituted benzofuran histamine H3 receptor antagonists : In vitro properties, drug-likeness, and behavioral activity |
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