COMBINATORIAL PROCESS FOR SYNTHESIZING AZETIDINONE ANALOGS

This invention relates to libraries of azetidinone peptide-like compounds and a combinatorial process for synthesis. Selected compounds are biologically active as inhibitors of the Vasopressin (V1a) receptor. La présente invention concerne d'une part des banques de composés d'azétidinone d...

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Bibliographic Details
Main Authors SKELTON, JEFFREY, J, BRUNS, ROBERT, F, CHANEY, MICHAEL, O, KOPPEL, GARY, A, COOPER, ROBIN, D., G, HUNDEN, DAVID, C
Format Patent
LanguageEnglish
French
Published 07.11.1996
Edition6
Subjects
APPARATUS THEREFOR
CHEMISTRY
COMBINATORIAL CHEMISTRY
GENERAL METHODS OF ORGANIC CHEMISTRY
HETEROCYCLIC COMPOUNDS
LIBRARIES, e.g. CHEMICAL LIBRARIES, IN SILICOLIBRARIES
METALLURGY
ORGANIC CHEMISTRY
PEPTIDES
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Summary:This invention relates to libraries of azetidinone peptide-like compounds and a combinatorial process for synthesis. Selected compounds are biologically active as inhibitors of the Vasopressin (V1a) receptor. La présente invention concerne d'une part des banques de composés d'azétidinone de type peptide, et d'autre part un procédé combinatoire de synthèse. En l'occurrence, les composés sélectionnés sont biologiquement actifs en tant qu'inhibiteurs du récepteur de la de la Vasopressine (V1a).
Bibliography:Application Number: WO1996US05397