NIRAPARIB SOLID STATE FORM
The present disclosure relates to a stabilized anhydrous p-toluenesulfonic acid salt of niraparib, Form A. The present disclosure is also related to processes for the preparation of the stabilized anhydrous p-toluenesulfonic acid salt of niraparib. Further, the present disclosure also relates to pha...
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| Format | Patent |
| Language | English French |
| Published |
09.04.2020
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| Abstract | The present disclosure relates to a stabilized anhydrous p-toluenesulfonic acid salt of niraparib, Form A. The present disclosure is also related to processes for the preparation of the stabilized anhydrous p-toluenesulfonic acid salt of niraparib. Further, the present disclosure also relates to pharmaceutical compositions comprising the stabilized anhydrous p-toluenesulfonic acid salt of niraparib and methods for treating disease using the stabilized anhydrous p-toluenesulfonic acid salt of niraparib.
La présente invention concerne un sel d'acide p-toluènesulfonique anhydre stabilisé de niraparib, forme A. Elle concerne également des procédés de préparation du sel d'acide p-toluènesulfonique anhydre stabilisé de niraparib. En outre, la présente invention concerne des compositions pharmaceutiques comprenant le sel d'acide p-toluènesulfonique anhydre stabilisé de niraparib et des procédés de traitement d'une maladie à l'aide du sel d'acide p-toluènesulfonique anhydre stabilisé de niraparib. |
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| AbstractList | The present disclosure relates to a stabilized anhydrous p-toluenesulfonic acid salt of niraparib, Form A. The present disclosure is also related to processes for the preparation of the stabilized anhydrous p-toluenesulfonic acid salt of niraparib. Further, the present disclosure also relates to pharmaceutical compositions comprising the stabilized anhydrous p-toluenesulfonic acid salt of niraparib and methods for treating disease using the stabilized anhydrous p-toluenesulfonic acid salt of niraparib.
La présente invention concerne un sel d'acide p-toluènesulfonique anhydre stabilisé de niraparib, forme A. Elle concerne également des procédés de préparation du sel d'acide p-toluènesulfonique anhydre stabilisé de niraparib. En outre, la présente invention concerne des compositions pharmaceutiques comprenant le sel d'acide p-toluènesulfonique anhydre stabilisé de niraparib et des procédés de traitement d'une maladie à l'aide du sel d'acide p-toluènesulfonique anhydre stabilisé de niraparib. |
| Author | KAVURU, Padmini |
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| DocumentTitleAlternate | FORME SOLIDE DE NIRAPARIB |
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| RelatedCompanies | JOHNSON MATTHEY PUBLIC LIMITED COMPANY KAVURU, Padmini |
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| Snippet | The present disclosure relates to a stabilized anhydrous p-toluenesulfonic acid salt of niraparib, Form A. The present disclosure is also related to processes... |
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| Title | NIRAPARIB SOLID STATE FORM |
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