QUINAZOLINE DERIVATIVES USED AS INHIBITORS OF ERBB TYROSINE KINASE
A quinazoline derivative of the Formula (I): wherein the substituents are as defined in the text for use in the production of an anti proliferative effect which effect is produced alone or in part by inhibiting erbB2 receptor tyrosine kinase in a warm blooded animal such as man. L'invention con...
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Format | Patent |
Language | English French |
Published |
07.06.2007
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Abstract | A quinazoline derivative of the Formula (I): wherein the substituents are as defined in the text for use in the production of an anti proliferative effect which effect is produced alone or in part by inhibiting erbB2 receptor tyrosine kinase in a warm blooded animal such as man.
L'invention concerne un dérivé de quinazoline de formule (I), dans laquelle les substituants sont tels que définis dans la description. Ce dérivé est destiné à produire un effet antiprolifératif, cet effet étant produit uniquement ou partiellement par inhibition des tyrosine kinases erbB2 associées au récepteur chez un animal à sang chaud, notamment un humain. |
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AbstractList | A quinazoline derivative of the Formula (I): wherein the substituents are as defined in the text for use in the production of an anti proliferative effect which effect is produced alone or in part by inhibiting erbB2 receptor tyrosine kinase in a warm blooded animal such as man.
L'invention concerne un dérivé de quinazoline de formule (I), dans laquelle les substituants sont tels que définis dans la description. Ce dérivé est destiné à produire un effet antiprolifératif, cet effet étant produit uniquement ou partiellement par inhibition des tyrosine kinases erbB2 associées au récepteur chez un animal à sang chaud, notamment un humain. |
Author | BRADBURY, ROBERT, HUGH DUCRAY, RICHARD BARLAAM, BERNARD, CHRISTOPHE |
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DocumentTitleAlternate | DERIVES DE QUINAZOLINE UTILISES EN TANT QU'INHIBITEURS DES TYROSINE KINASES ERBB ASSOCIEES AU RECEPTEUR |
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Notes | Application Number: WO2006GB04451 |
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RelatedCompanies | BRADBURY, ROBERT, HUGH ASTRAZENECA UK LIMITED DUCRAY, RICHARD BARLAAM, BERNARD, CHRISTOPHE ASTRAZENECA AB |
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Snippet | A quinazoline derivative of the Formula (I): wherein the substituents are as defined in the text for use in the production of an anti proliferative effect... |
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SubjectTerms | CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS |
Title | QUINAZOLINE DERIVATIVES USED AS INHIBITORS OF ERBB TYROSINE KINASE |
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