INTERMEDIATE FOR PRODUCING CARBOXYPEPTIDASE B INHIBITOR

A compound represented by the general formula (1), a salt thereof, or a hydrate or solvate of either. These are intermediates for efficiently producing a phosphinic acid derivative which is a potent carboxypeptidase B inhibitor. (1) [In the formula, R and R may be the same or different and each inde...

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Main Authors KANEMOTO, KENICHI, FUSHIHARA, KENICHI, YONETA, TOSHIO, SUZUKI, KOKICHI
Format Patent
LanguageEnglish
French
Japanese
Published 29.04.2004
Edition7
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Abstract A compound represented by the general formula (1), a salt thereof, or a hydrate or solvate of either. These are intermediates for efficiently producing a phosphinic acid derivative which is a potent carboxypeptidase B inhibitor. (1) [In the formula, R and R may be the same or different and each independently represents hydrogen or an easily removable protective group; R represents hydrogen or an easily removable protective group; R represents hydrogen or an easily removable protective group; and m is an integer of 1 to 8.] L'invention concerne un composé représenté par la formule générale (1), un sel dudit composé ou un hydrate ou un solvate correspondant. Ces composés sont des produits intermédiaires permettant de produire efficacement un dérivé d'acide phosphinique constituant un puissant inhibiteur de la carboxypeptidase B. Dans ladite formule, R et R sont identiques ou différents et représentent chacun indépendamment hydrogène ou un groupe protecteur facilement supprimable, R représente hydrogène ou un groupe protecteur facilement supprimable, R représente hydrogène ou un groupe protecteur facilement supprimable, et m est un nombre entier compris entre 1 et 8.
AbstractList A compound represented by the general formula (1), a salt thereof, or a hydrate or solvate of either. These are intermediates for efficiently producing a phosphinic acid derivative which is a potent carboxypeptidase B inhibitor. (1) [In the formula, R and R may be the same or different and each independently represents hydrogen or an easily removable protective group; R represents hydrogen or an easily removable protective group; R represents hydrogen or an easily removable protective group; and m is an integer of 1 to 8.] L'invention concerne un composé représenté par la formule générale (1), un sel dudit composé ou un hydrate ou un solvate correspondant. Ces composés sont des produits intermédiaires permettant de produire efficacement un dérivé d'acide phosphinique constituant un puissant inhibiteur de la carboxypeptidase B. Dans ladite formule, R et R sont identiques ou différents et représentent chacun indépendamment hydrogène ou un groupe protecteur facilement supprimable, R représente hydrogène ou un groupe protecteur facilement supprimable, R représente hydrogène ou un groupe protecteur facilement supprimable, et m est un nombre entier compris entre 1 et 8.
Author SUZUKI, KOKICHI
FUSHIHARA, KENICHI
KANEMOTO, KENICHI
YONETA, TOSHIO
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DocumentTitleAlternate PRODUIT INTERMEDIAIRE POUR LA PRODUCTION D'UN INHIBITEUR DE LA CARBOXYPEPTIDASE B
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RelatedCompanies SUZUKI, KOKICHI
FUSHIHARA, KENICHI
MEIJI SEIKA KAISHA, LTD
KANEMOTO, KENICHI
YONETA, TOSHIO
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Snippet A compound represented by the general formula (1), a salt thereof, or a hydrate or solvate of either. These are intermediates for efficiently producing a...
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SubjectTerms ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAININGELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN,SULFUR, SELENIUM OR TELLURIUM
CHEMISTRY
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
Title INTERMEDIATE FOR PRODUCING CARBOXYPEPTIDASE B INHIBITOR
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