Pyridone derivatives as acid secretion inhibitors and process for preparation thereof

The present invention relates to the preparation of stable pyridone disulphide derivatives having general formula (I) and its stereoisomers, which are useful in the treatment of gastrointestinal disorders. Pyridone disulphide derivatives (I) wherein, R1, R2 and R3 are independently alkyl, alkoxy, ha...

Full description

Saved in:
Bibliographic Details
Main Authors Tripathy Narendra Kumar, Chaudhari Ashok Tukaram, Mehta Samit Satish, Mahale Rajendra Dagesing, Gurjar Mukund Keshav, Pawar Sanjay Shankar, Kalhapure Vijay Keshav, Maikap Golakchandra Sudarshan, Khaladkar Tushar Pandurang
Format Patent
LanguageEnglish
Published 20.09.2016
Subjects
CHEMISTRY
HETEROCYCLIC COMPOUNDS
METALLURGY
ORGANIC CHEMISTRY
Online AccessGet full text

Cover

Abstract The present invention relates to the preparation of stable pyridone disulphide derivatives having general formula (I) and its stereoisomers, which are useful in the treatment of gastrointestinal disorders. Pyridone disulphide derivatives (I) wherein, R1, R2 and R3 are independently alkyl, alkoxy, halogen, halogenated alkoxy, halogenated alkyl, hydrogen and could be the same or different and X is CH or N. R1 is methyl, methoxy, fluorine, trifluoromethyl, difluoromethoxy and hydrogen, R2 is methyl, methoxy and hydrogen, and R3 is methyl and hydrogen.
AbstractList The present invention relates to the preparation of stable pyridone disulphide derivatives having general formula (I) and its stereoisomers, which are useful in the treatment of gastrointestinal disorders. Pyridone disulphide derivatives (I) wherein, R1, R2 and R3 are independently alkyl, alkoxy, halogen, halogenated alkoxy, halogenated alkyl, hydrogen and could be the same or different and X is CH or N. R1 is methyl, methoxy, fluorine, trifluoromethyl, difluoromethoxy and hydrogen, R2 is methyl, methoxy and hydrogen, and R3 is methyl and hydrogen.
Author Tripathy Narendra Kumar
Gurjar Mukund Keshav
Maikap Golakchandra Sudarshan
Mehta Samit Satish
Chaudhari Ashok Tukaram
Pawar Sanjay Shankar
Mahale Rajendra Dagesing
Khaladkar Tushar Pandurang
Kalhapure Vijay Keshav
Author_xml – fullname: Tripathy Narendra Kumar
– fullname: Chaudhari Ashok Tukaram
– fullname: Mehta Samit Satish
– fullname: Mahale Rajendra Dagesing
– fullname: Gurjar Mukund Keshav
– fullname: Pawar Sanjay Shankar
– fullname: Kalhapure Vijay Keshav
– fullname: Maikap Golakchandra Sudarshan
– fullname: Khaladkar Tushar Pandurang
BookMark eNqNiksKAjEQBbPQhb879AUE0QGZraK4FHTWQ0xemIYhHTphwNsbxAMID15B1dLMokQsTHd_K_uK5KE82cITMtk6x54ynKKwROI48IuLaDXRU1JxyJmCaGUkq_ablQEKCWszD3bM2Px-Zeh6eZ5vWyTpkZN1iCh992ib5rhrm9P-8EfyAf_WO30
ContentType Patent
DBID EVB
DatabaseName esp@cenet
DatabaseTitleList
Database_xml – sequence: 1
  dbid: EVB
  name: esp@cenet
  url: http://worldwide.espacenet.com/singleLineSearch?locale=en_EP
  sourceTypes: Open Access Repository
DeliveryMethod fulltext_linktorsrc
Discipline Medicine
Chemistry
Sciences
ExternalDocumentID US9447094B2
GroupedDBID EVB
ID FETCH-epo_espacenet_US9447094B23
IEDL.DBID EVB
IngestDate Fri Jul 19 14:55:16 EDT 2024
IsOpenAccess true
IsPeerReviewed false
IsScholarly false
Language English
LinkModel DirectLink
MergedId FETCHMERGED-epo_espacenet_US9447094B23
Notes Application Number: US201514703515
OpenAccessLink https://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20160920&DB=EPODOC&CC=US&NR=9447094B2
ParticipantIDs epo_espacenet_US9447094B2
PublicationCentury 2000
PublicationDate 20160920
PublicationDateYYYYMMDD 2016-09-20
PublicationDate_xml – month: 09
  year: 2016
  text: 20160920
  day: 20
PublicationDecade 2010
PublicationYear 2016
RelatedCompanies Emcure Pharmaceuticals Limited
RelatedCompanies_xml – name: Emcure Pharmaceuticals Limited
Score 3.0587106
Snippet The present invention relates to the preparation of stable pyridone disulphide derivatives having general formula (I) and its stereoisomers, which are useful...
SourceID epo
SourceType Open Access Repository
SubjectTerms CHEMISTRY
HETEROCYCLIC COMPOUNDS
METALLURGY
ORGANIC CHEMISTRY
Title Pyridone derivatives as acid secretion inhibitors and process for preparation thereof
URI https://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20160920&DB=EPODOC&locale=&CC=US&NR=9447094B2
hasFullText 1
inHoldings 1
isFullTextHit
isPrint
link http://utb.summon.serialssolutions.com/2.0.0/link/0/eLvHCXMwfV3dS8MwED_GFPVNp-L8Ig_St2HTZVvzUIS1G0PYB26VvY2mSTEvXVmr4n_vpeumLwp5OJKQjyOX3CV3vwA8oIXgUluiWRJRc1uleIsrwVpO7EqVxJFgiXnRHU-6o5A9LzvLGuhdLEyJE_pZgiOiRMUo70W5X2c_l1hB6VuZPwqNWeun4cILrMo6pl2bO7YV9L3BbBpMfcv3vXBuTV48zlgPLZk-7tYHRos2MPuD174JSsl-nyjDUzicYWNpcQY1lTbg2N99vNaAo3H13o1kJXr5OYSzr42W61QRiYvmo8TrzkmEKdaS5Eb7M8MmOn3TQps_dEiUSpJtAwEI6qZIqy3SN1Yzep9aJxdAhoOFP2rh-FZ7XqzC-X4m7Uuop9jtFRCHy3YsqHCidsIE7bqi06Ocq9iNGJWCNaH5ZzPX_5TdwIlhqvGPcOxbqBebd3WHh3Ah7kv2fQPqJo7D
link.rule.ids 230,309,786,891,25594,76903
linkProvider European Patent Office
linkToHtml http://utb.summon.serialssolutions.com/2.0.0/link/0/eLvHCXMwfV1LT8MwDLamgRg3GCDGMwfU20TbZV1zqJDWbhqwl9iKdpuaJhW9dNNaQPx7nOwBF5ByiJIoDyt2_DmxA3CHCMG1TIGwJLKUtUqyOpOc1u3YFTKJI04TdaM7GDq9kD7NmrMSpFtfGB0n9FMHR0SOipHfCy2vlz9GrEC_rczveYpFi4fu1AuMDTq2HJPZphG0vc54FIx8w_e9cGIMXzxGaQuRTBul9V4LEaFGSq9t5ZSy_H2idI9gf4ydZcUxlGRWhYq__XitCgeDzX03Zjesl59AOP5apWKRSSJw03zoeN05iTDFqSC50v7UtEmavaU8VX_okCgTZLl2BCCom2JeriN9YzOl98lFcgqk25n6vTrOb76jxTyc7FbSOINyhsOeA7GZaMTc4nbUSCi3HJc3WxZjMnYjaglOa1D7s5uLf-puodKbDvrz_uPw-RIOFYHVWwnbvIJysXqX13ggF_xGk_IbvF-RrQ
openUrl ctx_ver=Z39.88-2004&ctx_enc=info%3Aofi%2Fenc%3AUTF-8&rfr_id=info%3Asid%2Fsummon.serialssolutions.com&rft_val_fmt=info%3Aofi%2Ffmt%3Akev%3Amtx%3Apatent&rft.title=Pyridone+derivatives+as+acid+secretion+inhibitors+and+process+for+preparation+thereof&rft.inventor=Tripathy+Narendra+Kumar&rft.inventor=Chaudhari+Ashok+Tukaram&rft.inventor=Mehta+Samit+Satish&rft.inventor=Mahale+Rajendra+Dagesing&rft.inventor=Gurjar+Mukund+Keshav&rft.inventor=Pawar+Sanjay+Shankar&rft.inventor=Kalhapure+Vijay+Keshav&rft.inventor=Maikap+Golakchandra+Sudarshan&rft.inventor=Khaladkar+Tushar+Pandurang&rft.date=2016-09-20&rft.externalDBID=B2&rft.externalDocID=US9447094B2