Processes for the preparation of 5-HT2C receptor agonists

The present invention relates to processes and intermediates useful in the preparation of (R)-8-chloro-1-methyl-2,3,4,5-tetrahydro-1H-3-benzazepine (lorcaserin), a serotonin (5-HT) receptor modulator that is useful in the treatment of for example, central nervous system disorders, such as obesity.

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Bibliographic Details
Main Authors SHAW STEPHEN M, MACIAS MARK, LU XIAO-XIONG, CASTRO RYAN O, CHUANG TSUNG-HSUN, MARLON CARLOS, HADD MARK ALLEN, DEMATTEI JOHN A
Format Patent
LanguageEnglish
Published 10.02.2015
Subjects
ACYCLIC OR CARBOCYCLIC COMPOUNDS
CHEMISTRY
METALLURGY
ORGANIC CHEMISTRY
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Summary:The present invention relates to processes and intermediates useful in the preparation of (R)-8-chloro-1-methyl-2,3,4,5-tetrahydro-1H-3-benzazepine (lorcaserin), a serotonin (5-HT) receptor modulator that is useful in the treatment of for example, central nervous system disorders, such as obesity.
Bibliography:Application Number: US201013378797