Substituted thiazolo[3,2-a]azepine derivatives

The present invention relates to a substituted thiazolo[3,2-a] azepine derivative having inhibitory activity against angiotensin I converting enzyme and neutral endpeptidase and is represented by the following general formula (I):

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Main Authors MATSUOKA; TOSHIYUKI, MIZUNO; MASANORI, SAITO; MAMORU, ADACHI; HIDEYUKI, OKITA; MAKOTO, MATSUSHIMA; TOMOHIRO, OINUMA; HITOSHI, NAMIKI; MASAYUKI, YONEDA; NAOKI, SUDO; TAKESHI, KOTAKE; MAKOTO, MIYAKE; KAZUTOSHI, FUKUDA; YOSHIO, SUDA; SHINJI
Format Patent
LanguageEnglish
Published 18.04.2000
Edition7
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Abstract The present invention relates to a substituted thiazolo[3,2-a] azepine derivative having inhibitory activity against angiotensin I converting enzyme and neutral endpeptidase and is represented by the following general formula (I):
AbstractList The present invention relates to a substituted thiazolo[3,2-a] azepine derivative having inhibitory activity against angiotensin I converting enzyme and neutral endpeptidase and is represented by the following general formula (I):
Author KOTAKE; MAKOTO
OKITA; MAKOTO
FUKUDA; YOSHIO
NAMIKI; MASAYUKI
MATSUOKA; TOSHIYUKI
YONEDA; NAOKI
SUDA; SHINJI
MIYAKE; KAZUTOSHI
OINUMA; HITOSHI
MIZUNO; MASANORI
ADACHI; HIDEYUKI
SUDO; TAKESHI
SAITO; MAMORU
MATSUSHIMA; TOMOHIRO
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– fullname: OINUMA; HITOSHI
– fullname: NAMIKI; MASAYUKI
– fullname: YONEDA; NAOKI
– fullname: SUDO; TAKESHI
– fullname: KOTAKE; MAKOTO
– fullname: MIYAKE; KAZUTOSHI
– fullname: FUKUDA; YOSHIO
– fullname: SUDA; SHINJI
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Snippet The present invention relates to a substituted thiazolo[3,2-a] azepine derivative having inhibitory activity against angiotensin I converting enzyme and...
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SubjectTerms CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PEPTIDES
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
Title Substituted thiazolo[3,2-a]azepine derivatives
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