Preparation of 2-(2'-thienyl)ethylamine derivatives and synthesis of thieno[3,2-c]pyridine derivatives therefrom
An improved process for the synthesis of 2-(2'-thienyl)ethylamine from suitably functionalized derivatives of 2-(2'-thienyl)ethanol employing ammonia gas in the presence of a metal salt or liquid ammonia and alkyl ketone as a solvent. The 2-(2'-thienyl)ethylamine produced by this proc...
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| Main Author | |
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| Format | Patent |
| Language | English |
| Published |
02.03.1993
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| Subjects | |
| Online Access | Get full text |
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| Abstract | An improved process for the synthesis of 2-(2'-thienyl)ethylamine from suitably functionalized derivatives of 2-(2'-thienyl)ethanol employing ammonia gas in the presence of a metal salt or liquid ammonia and alkyl ketone as a solvent. The 2-(2'-thienyl)ethylamine produced by this process is advantageously converted to ticlopidine. |
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| AbstractList | An improved process for the synthesis of 2-(2'-thienyl)ethylamine from suitably functionalized derivatives of 2-(2'-thienyl)ethanol employing ammonia gas in the presence of a metal salt or liquid ammonia and alkyl ketone as a solvent. The 2-(2'-thienyl)ethylamine produced by this process is advantageously converted to ticlopidine. |
| Author | DEHOFF; BRADLEY S |
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| Notes | Application Number: US19910738697 |
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| PublicationDateYYYYMMDD | 1993-03-02 |
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| PublicationDecade | 1990 |
| PublicationYear | 1993 |
| RelatedCompanies | SYNTEX (U.S.A.) INC |
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| Title | Preparation of 2-(2'-thienyl)ethylamine derivatives and synthesis of thieno[3,2-c]pyridine derivatives therefrom |
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