Pyrazolone-Fused Pyrimidine Compound, and Preparation Method and Use Therefor

Disclosed in the present invention are a pyrazolone-fused pyrimidine compound, and a preparation method and a use therefor. Provided in the present invention is a pyrazolone-fused pyrimidine compound as in formula (I), said compound having better inhibitory activity towards WEE1 kinase.

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Main Authors YU, Jianxin, GE, Hui, ZHANG, Zhihui, XIA, Guangxin, SHU, Sijie, ZHANG, Bingbin, SHI, Chen, KE, Ying, LIU, Yanjun, LOU, Jiangsong, HUO, Guoyong, WANG, Qian, MAO, Yu, ZHANG, Chi, ZHANG, Lin
Format Patent
LanguageEnglish
Published 13.10.2022
Subjects
CHEMISTRY
HETEROCYCLIC COMPOUNDS
METALLURGY
ORGANIC CHEMISTRY
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Abstract Disclosed in the present invention are a pyrazolone-fused pyrimidine compound, and a preparation method and a use therefor. Provided in the present invention is a pyrazolone-fused pyrimidine compound as in formula (I), said compound having better inhibitory activity towards WEE1 kinase.
AbstractList Disclosed in the present invention are a pyrazolone-fused pyrimidine compound, and a preparation method and a use therefor. Provided in the present invention is a pyrazolone-fused pyrimidine compound as in formula (I), said compound having better inhibitory activity towards WEE1 kinase.
Author ZHANG, Chi
ZHANG, Zhihui
ZHANG, Bingbin
MAO, Yu
YU, Jianxin
HUO, Guoyong
SHI, Chen
WANG, Qian
ZHANG, Lin
XIA, Guangxin
LOU, Jiangsong
LIU, Yanjun
GE, Hui
SHU, Sijie
KE, Ying
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– fullname: ZHANG, Bingbin
– fullname: SHI, Chen
– fullname: KE, Ying
– fullname: LIU, Yanjun
– fullname: LOU, Jiangsong
– fullname: HUO, Guoyong
– fullname: WANG, Qian
– fullname: MAO, Yu
– fullname: ZHANG, Chi
– fullname: ZHANG, Lin
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Snippet Disclosed in the present invention are a pyrazolone-fused pyrimidine compound, and a preparation method and a use therefor. Provided in the present invention...
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HETEROCYCLIC COMPOUNDS
METALLURGY
ORGANIC CHEMISTRY
Title Pyrazolone-Fused Pyrimidine Compound, and Preparation Method and Use Therefor
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