SPIROHEPTANYL HYDANTOINS AS ROCK INHIBITORS
The present invention provides compounds of Formula (I): or stereoisomers, tautomers, or pharmaceutically acceptable salts thereof, wherein all the variables are as defined herein. These compounds are selective ROCK inhibitors. This invention also relates to pharmaceutical compositions comprising th...
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| Main Authors | , |
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| Format | Patent |
| Language | English |
| Published |
27.05.2021
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| Subjects | |
| Online Access | Get full text |
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| Abstract | The present invention provides compounds of Formula (I): or stereoisomers, tautomers, or pharmaceutically acceptable salts thereof, wherein all the variables are as defined herein. These compounds are selective ROCK inhibitors. This invention also relates to pharmaceutical compositions comprising these compounds and methods of treating cardiovascular, smooth muscle, oncologic, neuropathologic, autoimmune, fibrotic, and/or inflammatory disorders using the same. |
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| AbstractList | The present invention provides compounds of Formula (I): or stereoisomers, tautomers, or pharmaceutically acceptable salts thereof, wherein all the variables are as defined herein. These compounds are selective ROCK inhibitors. This invention also relates to pharmaceutical compositions comprising these compounds and methods of treating cardiovascular, smooth muscle, oncologic, neuropathologic, autoimmune, fibrotic, and/or inflammatory disorders using the same. |
| Author | Shaw, Scott A Vokits, Benjamin P |
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| RelatedCompanies | BRISTOL-MYERS SQUIBB COMPANY |
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| Snippet | The present invention provides compounds of Formula (I): or stereoisomers, tautomers, or pharmaceutically acceptable salts thereof, wherein all the variables... |
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| Title | SPIROHEPTANYL HYDANTOINS AS ROCK INHIBITORS |
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