Peripheral Opioid Receptor Antagonists and Uses Thereof

The present invention provides a compound of formula I: wherein X−, R1, and R2 are as defined herein, and compositions thereof.

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Main Authors SZELIGA JAN, FABIAN STEVEN R, SHAH SYED M, BAZHINA NATALIYA, OFSLAGER CHRISTIAN, LOKHNAUTH JOHN, MEGATI SREENIVASULU, RADEBAUGH GALEN, MELUCCI CHARLES, DONATO, III GEORGE JOSEPH, ZHANG HUYI, PATEL NIKETA, ZHU TIANMIN
Format Patent
LanguageEnglish
Published 13.12.2012
Subjects
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
Online AccessGet full text

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Abstract The present invention provides a compound of formula I: wherein X−, R1, and R2 are as defined herein, and compositions thereof.
AbstractList The present invention provides a compound of formula I: wherein X−, R1, and R2 are as defined herein, and compositions thereof.
Author ZHANG HUYI
LOKHNAUTH JOHN
MEGATI SREENIVASULU
SHAH SYED M
DONATO, III GEORGE JOSEPH
RADEBAUGH GALEN
MELUCCI CHARLES
ZHU TIANMIN
FABIAN STEVEN R
OFSLAGER CHRISTIAN
SZELIGA JAN
PATEL NIKETA
BAZHINA NATALIYA
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– fullname: LOKHNAUTH JOHN
– fullname: MEGATI SREENIVASULU
– fullname: RADEBAUGH GALEN
– fullname: MELUCCI CHARLES
– fullname: DONATO, III GEORGE JOSEPH
– fullname: ZHANG HUYI
– fullname: PATEL NIKETA
– fullname: ZHU TIANMIN
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SHAH SYED M
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BAZHINA NATALIYA
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Snippet The present invention provides a compound of formula I: wherein X−, R1, and R2 are as defined herein, and compositions thereof.
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HYGIENE
MEDICAL OR VETERINARY SCIENCE
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
Title Peripheral Opioid Receptor Antagonists and Uses Thereof
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