Thienopyrroles as histone demethylase inhibitors

• Main Authors: Meroni, Giuseppe, Mercurio, Ciro, Romussi, Alessia, Varasi, Mario, Moretti, Loris, Zagarri, Elisa, Vianello, Paola, Cappa, Anna, Villa, Manuela, Sartori, Luca
• Format: Patent
• Language: English
• Published: 22.01.2019
• Subjects: CHEMISTRY; HETEROCYCLIC COMPOUNDS; HUMAN NECESSITIES; HYGIENE; MEDICAL OR VETERINARY SCIENCE; METALLURGY; ORGANIC CHEMISTRY; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES

The present invention relates to thienopyrrole derivatives, wherein R, R 1 , R 2 and R 3 are as defined in the specification, pharmaceutical compositions containing such compounds and to their use in therapy.