MK2 inhibitors, the synthesis thereof, and intermediates thereto

The present disclosure provides novel synthetic intermediates useful in the synthesis of MK2 kinase inhibitors.

Saved in:
Bibliographic Details
Main Authors COOMBS, JOHN R, LIM, DANIEL, ZHU, KEMING, GEORGE, DAVID T, RUCHELMAN, ALEXANDER L, LIN, DONG, JOE, CANDICE LEE, ZHENG, BIN
Format Patent
LanguageChinese
English
Published 01.12.2022
Subjects
Online AccessGet full text

Cover

Loading…
Abstract The present disclosure provides novel synthetic intermediates useful in the synthesis of MK2 kinase inhibitors.
AbstractList The present disclosure provides novel synthetic intermediates useful in the synthesis of MK2 kinase inhibitors.
Author ZHU, KEMING
ZHENG, BIN
LIM, DANIEL
LIN, DONG
RUCHELMAN, ALEXANDER L
JOE, CANDICE LEE
COOMBS, JOHN R
GEORGE, DAVID T
Author_xml – fullname: COOMBS, JOHN R
– fullname: LIM, DANIEL
– fullname: ZHU, KEMING
– fullname: GEORGE, DAVID T
– fullname: RUCHELMAN, ALEXANDER L
– fullname: LIN, DONG
– fullname: JOE, CANDICE LEE
– fullname: ZHENG, BIN
BookMark eNrjYmDJy89L5WRw8PU2UsjMy8hMyizJLyrWUSjJSFUorswDUsWZxSBeUWp-mo5CYl4KUFlJalFuakpmYkkqVKokn4eBNS0xpziVF0pzMyi6uYY4e-imFuTHpxYXJCan5qWWxIeEGxkYGZmYGVkYORoTowYAt_IzAg
ContentType Patent
DBID EVB
DatabaseName esp@cenet
DatabaseTitleList
Database_xml – sequence: 1
  dbid: EVB
  name: esp@cenet
  url: http://worldwide.espacenet.com/singleLineSearch?locale=en_EP
  sourceTypes: Open Access Repository
DeliveryMethod fulltext_linktorsrc
Discipline Medicine
Chemistry
Sciences
ExternalDocumentID TW202246282A
GroupedDBID EVB
ID FETCH-epo_espacenet_TW202246282A3
IEDL.DBID EVB
IngestDate Fri Aug 09 05:00:59 EDT 2024
IsOpenAccess true
IsPeerReviewed false
IsScholarly false
Language Chinese
English
LinkModel DirectLink
MergedId FETCHMERGED-epo_espacenet_TW202246282A3
Notes Application Number: TW202211104117
OpenAccessLink https://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20221201&DB=EPODOC&CC=TW&NR=202246282A
ParticipantIDs epo_espacenet_TW202246282A
PublicationCentury 2000
PublicationDate 20221201
PublicationDateYYYYMMDD 2022-12-01
PublicationDate_xml – month: 12
  year: 2022
  text: 20221201
  day: 01
PublicationDecade 2020
PublicationYear 2022
RelatedCompanies CELGENE CORPORATION
RelatedCompanies_xml – name: CELGENE CORPORATION
Score 3.550453
Snippet The present disclosure provides novel synthetic intermediates useful in the synthesis of MK2 kinase inhibitors.
SourceID epo
SourceType Open Access Repository
SubjectTerms CHEMISTRY
HETEROCYCLIC COMPOUNDS
METALLURGY
ORGANIC CHEMISTRY
Title MK2 inhibitors, the synthesis thereof, and intermediates thereto
URI https://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20221201&DB=EPODOC&locale=&CC=TW&NR=202246282A
hasFullText 1
inHoldings 1
isFullTextHit
isPrint
link http://utb.summon.serialssolutions.com/2.0.0/link/0/eLvHCXMwY2BQAe2uNjM3S9YF4hRdE4s0A90kU2CEmFkkG5omp5glp4H3cfv6mXmEmnhFmEYwMWTB9sKAzwktBx-OCMxRycD8XgIurwsQg1gu4LWVxfpJmUChfHu3EFsXNWjv2AhYEAP7xi5Otq4B_i7-zmrOzrYh4Wp-QWA50DZMI0dmBlZQMxp0zr5rmBNoV0oBcpXiJsjAFgA0La9EiIGpKkOYgdMZdvOaMAOHL3TCG8iE5r1iEQYHX28jhcy8jMykTNANOToKwKabQnFlHpAqziwG8YpS89N0FBLzUhRAh0AUgTeFAFuSEKmSfFEGRTfXEGcPXaBT4uH-jg8JR7jaWIyBJS8_L1WCQSHJEtgbNk9KS7VISjRJMbRMtEgE9S2BGdc4LdHC2FCSQQq3OVL4JKUZuEAcyGoNGQaWkqLSVFlgnVuSJAcOLABcJ4YN
link.rule.ids 230,309,786,891,25594,76906
linkProvider European Patent Office
linkToHtml http://utb.summon.serialssolutions.com/2.0.0/link/0/eLvHCXMwY2BQAe2uNjM3S9YF4hRdE4s0A90kU2CEmFkkG5omp5glp4H3cfv6mXmEmnhFmEYwMWTB9sKAzwktBx-OCMxRycD8XgIurwsQg1gu4LWVxfpJmUChfHu3EFsXNWjv2AhYEAP7xi5Otq4B_i7-zmrOzrYh4Wp-QWA50DZMI0dmBlZz0Om8oKZTmBNoV0oBcpXiJsjAFgA0La9EiIGpKkOYgdMZdvOaMAOHL3TCG8iE5r1iEQYHX28jhcy8jMykTNANOToKwKabQnFlHpAqziwG8YpS89N0FBLzUhRAh0AUgTeFAFuSEKmSfFEGRTfXEGcPXaBT4uH-jg8JR7jaWIyBJS8_L1WCQSHJEtgbNk9KS7VISjRJMbRMtEgE9S2BGdc4LdHC2FCSQQq3OVL4JOUZOD1CfH3ifTz9vKUZuEASkJUbMgwsJUWlqbLA-rckSQ4ccADKAYj6
openUrl ctx_ver=Z39.88-2004&ctx_enc=info%3Aofi%2Fenc%3AUTF-8&rfr_id=info%3Asid%2Fsummon.serialssolutions.com&rft_val_fmt=info%3Aofi%2Ffmt%3Akev%3Amtx%3Apatent&rft.title=MK2+inhibitors%2C+the+synthesis+thereof%2C+and+intermediates+thereto&rft.inventor=COOMBS%2C+JOHN+R&rft.inventor=LIM%2C+DANIEL&rft.inventor=ZHU%2C+KEMING&rft.inventor=GEORGE%2C+DAVID+T&rft.inventor=RUCHELMAN%2C+ALEXANDER+L&rft.inventor=LIN%2C+DONG&rft.inventor=JOE%2C+CANDICE+LEE&rft.inventor=ZHENG%2C+BIN&rft.date=2022-12-01&rft.externalDBID=A&rft.externalDocID=TW202246282A