Azabicyclic heterocycles as cannabinoid receptor modulators

The present application describes compounds according to Formula I, pharmaceutical compositions comprising at least one compound according to Formula I and optionally one or more additional therapeutic agents and methods of treatment using the compounds according to Formula I both alone and in combi...

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Main Authors SUN, CHONG-QING, WU, XIMAO, ELLSWORTH, BRUCE, EWING, WILLIAM R, GU, ZHENGXIANG, JOHNSON, STEPHEN R, YU, GUI-XUE, GERRITZ, SAMUEL W, WU, GANG, HUANG, YAN-TING, SHER, PHILIP M, PENDRI, ANNAPURNA, SITKOFF, DOREE F, WANG, YING, MIKKILINENI, AMARENDRA B, MURUGESAN, NATESAN
Format Patent
LanguageChinese
English
Published 01.09.2005
Subjects
CHEMISTRY
HETEROCYCLIC COMPOUNDS
METALLURGY
ORGANIC CHEMISTRY
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Abstract The present application describes compounds according to Formula I, pharmaceutical compositions comprising at least one compound according to Formula I and optionally one or more additional therapeutic agents and methods of treatment using the compounds according to Formula I both alone and in combination with one or more additional therapeutic agents. The compounds have the general Formula I. , including all prodrugs, pharmaceutically acceptable salts and stereoisomers, R1, R2, R3, R6, R7, m and n are described herein:
AbstractList The present application describes compounds according to Formula I, pharmaceutical compositions comprising at least one compound according to Formula I and optionally one or more additional therapeutic agents and methods of treatment using the compounds according to Formula I both alone and in combination with one or more additional therapeutic agents. The compounds have the general Formula I. , including all prodrugs, pharmaceutically acceptable salts and stereoisomers, R1, R2, R3, R6, R7, m and n are described herein:
Author MURUGESAN, NATESAN
EWING, WILLIAM R
HUANG, YAN-TING
YU, GUI-XUE
PENDRI, ANNAPURNA
ELLSWORTH, BRUCE
WANG, YING
SUN, CHONG-QING
SITKOFF, DOREE F
SHER, PHILIP M
WU, GANG
WU, XIMAO
MIKKILINENI, AMARENDRA B
GU, ZHENGXIANG
JOHNSON, STEPHEN R
GERRITZ, SAMUEL W
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– fullname: YU, GUI-XUE
– fullname: GERRITZ, SAMUEL W
– fullname: WU, GANG
– fullname: HUANG, YAN-TING
– fullname: SHER, PHILIP M
– fullname: PENDRI, ANNAPURNA
– fullname: SITKOFF, DOREE F
– fullname: WANG, YING
– fullname: MIKKILINENI, AMARENDRA B
– fullname: MURUGESAN, NATESAN
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Snippet The present application describes compounds according to Formula I, pharmaceutical compositions comprising at least one compound according to Formula I and...
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SubjectTerms CHEMISTRY
HETEROCYCLIC COMPOUNDS
METALLURGY
ORGANIC CHEMISTRY
Title Azabicyclic heterocycles as cannabinoid receptor modulators
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