Processes and intermediates for the preparation of a pde10 inhibitor
Disclosed herein are (5-methyl-1,3,4-thiadiazol-2-yl)phenyl intermediates which are useful in the synthesis of the compound 1-(5-(4-chloro-3,5-dimethoxyphenyl)furan-2-yl)-2-ethoxy-2-(4-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl)ethanone, which is intended for use as a PDE10 inhibitor.
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Main Authors | , , , , , , , |
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Format | Patent |
Language | English |
Published |
28.07.2017
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Subjects | |
Online Access | Get full text |
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Abstract | Disclosed herein are (5-methyl-1,3,4-thiadiazol-2-yl)phenyl intermediates which are useful in the synthesis of the compound 1-(5-(4-chloro-3,5-dimethoxyphenyl)furan-2-yl)-2-ethoxy-2-(4-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl)ethanone, which is intended for use as a PDE10 inhibitor. |
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AbstractList | Disclosed herein are (5-methyl-1,3,4-thiadiazol-2-yl)phenyl intermediates which are useful in the synthesis of the compound 1-(5-(4-chloro-3,5-dimethoxyphenyl)furan-2-yl)-2-ethoxy-2-(4-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl)ethanone, which is intended for use as a PDE10 inhibitor. |
Author | Cutshall Neil S Mcdermott Michael James Luke Wayne Douglas Little Thomas L Gage Jennifer Lynn Brot Elisabeth C A Reineke Karl E Jonas Marco |
Author_xml | – fullname: Brot Elisabeth C A – fullname: Cutshall Neil S – fullname: Jonas Marco – fullname: Reineke Karl E – fullname: Gage Jennifer Lynn – fullname: Little Thomas L – fullname: Mcdermott Michael James – fullname: Luke Wayne Douglas |
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Title | Processes and intermediates for the preparation of a pde10 inhibitor |
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