N-(HETERO)ARYL-PYRROLIDINE DERIVATIVES OF PYRAZOL-4-YL-PYRROLO[2,3-D]PYRIMIDINES AND PYRROL-3-YL-PYRROLO[2,3-D]PYRIMIDINES AS JANUS KINASE INHIBITORS
THE PRESENT INVENTION RELATES TO N-(HETERO) ARYL-PYRROIIDIFLE DERIVATIVES OF FORMULA I, AS WELL AS THEIR COMPOSITIONS AND METHODS OF USE, WHICH ARE JAK INHIBITORS, SUCH AS SELECTIVE JAK1 INHIBITORS, USEFUL IN THE TREATMENT OF JAK-ASSOCIATED DISEASES INCLUDING, FOR EXAMPLE, INFLAMMATORY AND AUTOIMMUN...
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Format | Patent |
Language | English |
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15.03.2016
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Abstract | THE PRESENT INVENTION RELATES TO N-(HETERO) ARYL-PYRROIIDIFLE DERIVATIVES OF FORMULA I, AS WELL AS THEIR COMPOSITIONS AND METHODS OF USE, WHICH ARE JAK INHIBITORS, SUCH AS SELECTIVE JAK1 INHIBITORS, USEFUL IN THE TREATMENT OF JAK-ASSOCIATED DISEASES INCLUDING, FOR EXAMPLE, INFLAMMATORY AND AUTOIMMUNE DISORDERS, AS WELL AS CANCER. |
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AbstractList | THE PRESENT INVENTION RELATES TO N-(HETERO) ARYL-PYRROIIDIFLE DERIVATIVES OF FORMULA I, AS WELL AS THEIR COMPOSITIONS AND METHODS OF USE, WHICH ARE JAK INHIBITORS, SUCH AS SELECTIVE JAK1 INHIBITORS, USEFUL IN THE TREATMENT OF JAK-ASSOCIATED DISEASES INCLUDING, FOR EXAMPLE, INFLAMMATORY AND AUTOIMMUNE DISORDERS, AS WELL AS CANCER. |
Author | SHAO, LIXIN STORACE, LOUIS GLENN, JOSEPH P SHEPARD, STACEY ARVANITIS, ARGYRIOS G FOLMER, BEVERLY ZHU, WENYU RODGERS, JAMES D WANG, HAISHENG |
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Snippet | THE PRESENT INVENTION RELATES TO N-(HETERO) ARYL-PYRROIIDIFLE DERIVATIVES OF FORMULA I, AS WELL AS THEIR COMPOSITIONS AND METHODS OF USE, WHICH ARE JAK... |
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Title | N-(HETERO)ARYL-PYRROLIDINE DERIVATIVES OF PYRAZOL-4-YL-PYRROLO[2,3-D]PYRIMIDINES AND PYRROL-3-YL-PYRROLO[2,3-D]PYRIMIDINES AS JANUS KINASE INHIBITORS |
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