TRIAZOLOPYRIDINES AS PHOSPHODIESTERASE INHIBITORS FOR TREATMENT OF DERMAL DISEASES

The present invention relates to a compound according to formula I, wherein R1, R2 and A are as defined herein, which exhibit PDE4 inhibitory activity and may be used in the treatment of inflammatory diseases or autoimmune diseases, in particular inflammatory or proliferative dermal diseases. La pre...

Full description

Saved in:
Bibliographic Details
Main Authors ANNE MARIE HORNEMAN, THOMAS VIFIAN, SIMON FELDBAEK NIELSEN, JESPER FAERGEMANN LAU
Format Patent
LanguageEnglish
Spanish
Published 28.07.2011
Subjects
Online AccessGet full text

Cover

Loading…
Abstract The present invention relates to a compound according to formula I, wherein R1, R2 and A are as defined herein, which exhibit PDE4 inhibitory activity and may be used in the treatment of inflammatory diseases or autoimmune diseases, in particular inflammatory or proliferative dermal diseases. La presente invención se refiere a un compuesto de conformidad con la fórmula I, en donde R1, R2 y A son como se definen en la presente, el cual exhibe actividad inhibitoria de PDE4 y se pueden usar en el tratamiento de enfermedades inflamatorias o enfermedades autoinmunes, en particular enfermedades dérmicas inflamatorias o proliferativas. (Ver fórmula (I)).
AbstractList The present invention relates to a compound according to formula I, wherein R1, R2 and A are as defined herein, which exhibit PDE4 inhibitory activity and may be used in the treatment of inflammatory diseases or autoimmune diseases, in particular inflammatory or proliferative dermal diseases. La presente invención se refiere a un compuesto de conformidad con la fórmula I, en donde R1, R2 y A son como se definen en la presente, el cual exhibe actividad inhibitoria de PDE4 y se pueden usar en el tratamiento de enfermedades inflamatorias o enfermedades autoinmunes, en particular enfermedades dérmicas inflamatorias o proliferativas. (Ver fórmula (I)).
Author THOMAS VIFIAN
SIMON FELDBAEK NIELSEN
ANNE MARIE HORNEMAN
JESPER FAERGEMANN LAU
Author_xml – fullname: ANNE MARIE HORNEMAN
– fullname: THOMAS VIFIAN
– fullname: SIMON FELDBAEK NIELSEN
– fullname: JESPER FAERGEMANN LAU
BookMark eNqNyj0KwkAQQOEttPDvDoO9kMQgtqs7IQNJNsxMoTYhyFrJJhDvjyk8gMXjNd_aLOIQw8qwMtmHr3x7Z3LUoIAVaEsvc45QFNkKAjUlXUg9CxSeQRmt1tgo-AIccm0rcCQ4U9ma5at_T2H3-8bsC9RreQjj0IVp7J8hhk9X37IkTZPklGdne_wLfQHICzJr
ContentType Patent
DBID EVB
DatabaseName esp@cenet
DatabaseTitleList
Database_xml – sequence: 1
  dbid: EVB
  name: esp@cenet
  url: http://worldwide.espacenet.com/singleLineSearch?locale=en_EP
  sourceTypes: Open Access Repository
DeliveryMethod fulltext_linktorsrc
Discipline Medicine
Chemistry
Sciences
DocumentTitleAlternate TRIAZOLOPIRIDINAS COMO INHIBIDORES DE FOSFODIESTERASA PARA TRATAMIENTO DE ENFERMEDADES DERMICAS.
ExternalDocumentID MX2011006428A
GroupedDBID EVB
ID FETCH-epo_espacenet_MX2011006428A3
IEDL.DBID EVB
IngestDate Fri Jul 19 14:57:22 EDT 2024
IsOpenAccess true
IsPeerReviewed false
IsScholarly false
Language English
Spanish
LinkModel DirectLink
MergedId FETCHMERGED-epo_espacenet_MX2011006428A3
Notes Application Number: MX20110006428
OpenAccessLink https://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20110728&DB=EPODOC&CC=MX&NR=2011006428A
ParticipantIDs epo_espacenet_MX2011006428A
PublicationCentury 2000
PublicationDate 20110728
PublicationDateYYYYMMDD 2011-07-28
PublicationDate_xml – month: 07
  year: 2011
  text: 20110728
  day: 28
PublicationDecade 2010
PublicationYear 2011
RelatedCompanies LEO PHARMA A/S
RelatedCompanies_xml – name: LEO PHARMA A/S
Score 2.6898108
Snippet The present invention relates to a compound according to formula I, wherein R1, R2 and A are as defined herein, which exhibit PDE4 inhibitory activity and may...
SourceID epo
SourceType Open Access Repository
SubjectTerms CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
Title TRIAZOLOPYRIDINES AS PHOSPHODIESTERASE INHIBITORS FOR TREATMENT OF DERMAL DISEASES
URI https://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20110728&DB=EPODOC&locale=&CC=MX&NR=2011006428A
hasFullText 1
inHoldings 1
isFullTextHit
isPrint
link http://utb.summon.serialssolutions.com/2.0.0/link/0/eLvHCXMwfV1RS8MwED7mFPVNp6JOJYj0rbh1dV0fhnRNSivrUtIq1Zdh1wgibMNV_Pte4qZ72kMg5EJIAl_uy-XuAnDTRtagmLbZkhPHtJFhmwXyBBUFUlquVcqu9iaMR93w0X7I7_IafKxiYXSe0G-dHBERNUG8V_q8nv8bsaj2rVzcFu_YNLsPsj41ypW5r-VYPYMO-izhlPuG7_fj3BiJX5km294WbCOPdhQc2NNAhaXM13VKcAA7CQ43rQ6hJhcN2PNXX681YDdevnhjdQm-xRGITETeCx_y5FlEVP2WQbyUJCFPsShah8zUSxmJRmE0iDIuUoJXPJIJ5mUqZT_hAaFMxN6Q0Chl2DU9huuAZX5o4uTGf1sxjvO1hXROoD6dTeUpkE6JK--6dtnuOLZbSFe2ilcXsVk4b267nJxBc8NA5xulTdj_NaQ6ptW7gHr1-SUvURNXxZXewR82sYSd
link.rule.ids 230,309,783,888,25576,76876
linkProvider European Patent Office
linkToHtml http://utb.summon.serialssolutions.com/2.0.0/link/0/eLvHCXMwfV3dS8MwED_mFOebTkWdH0Gkb8Wtq-v6MKTrB622TUmjVF-GXSOIsA1X8d_30m26pz0EQi6EJPDL_XK5uwDcdJA1SKattsXYUHVk2GqOPEFGgRSaqRWiV3kTRnHPf9IfsrusBp-rWJgqT-hPlRwRETVGvJfVeT37N2I5lW_l_Db_wKbpvccHjlKszH1tQ-srznDgJtShtmLbgyhTYraQVWTb2oJt5NiGhIP7PJRhKbN1neLtw06Cw03KA6iJeRMa9urrtSbsRssXb6wuwTc_BMZZYL3SkCYvLHDkbxnESkni0xSLpHXITK3UJUHsB8OAU5YSvOIRzlyLy5T9hHrEcVlkhcQJUhe7pkdw7bnc9lWc3OhvK0ZRtraQ7jHUJ9OJOAHSLXDlPVMvOl1DN3Nhinb-ZiI2c-Pd7BTjU2htGOhso_QKGj6PwlEYxI8t2FsYVQ1V659Dvfz6Fheolcv8strNX5sLh5A
openUrl ctx_ver=Z39.88-2004&ctx_enc=info%3Aofi%2Fenc%3AUTF-8&rfr_id=info%3Asid%2Fsummon.serialssolutions.com&rft_val_fmt=info%3Aofi%2Ffmt%3Akev%3Amtx%3Apatent&rft.title=TRIAZOLOPYRIDINES+AS+PHOSPHODIESTERASE+INHIBITORS+FOR+TREATMENT+OF+DERMAL+DISEASES&rft.inventor=ANNE+MARIE+HORNEMAN&rft.inventor=THOMAS+VIFIAN&rft.inventor=SIMON+FELDBAEK+NIELSEN&rft.inventor=JESPER+FAERGEMANN+LAU&rft.date=2011-07-28&rft.externalDBID=A&rft.externalDocID=MX2011006428A