단백질 키나제 저해제로서 유용한 피리도퀴나졸린의 카르복시산 유도체
본 발명은 단백질 키나제의 강력한 저해제로서 11-옥소-11H-피리도 [2,1-b]퀴나졸린-6-카르복사미드의 신규한 카르복시산 유도체, 이를 포함하는 약학적 조성물, 및 단백질 키나제를 저해함으로써 개선할 수 있는 질환 또는 병리학적 질환을 치료하기 위한 약제의 제조에 있어 상기한 화합물의 용도에 관한 것이다. The present invention relates to novel carboxylic acid derivatives of 11-oxo-11H-pyrido [2,1-b]quinazoline-6-carboxamide as p...
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| Main Authors | , |
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| Format | Patent |
| Language | Korean |
| Published |
05.02.2020
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| Subjects | |
| Online Access | Get full text |
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| Abstract | 본 발명은 단백질 키나제의 강력한 저해제로서 11-옥소-11H-피리도 [2,1-b]퀴나졸린-6-카르복사미드의 신규한 카르복시산 유도체, 이를 포함하는 약학적 조성물, 및 단백질 키나제를 저해함으로써 개선할 수 있는 질환 또는 병리학적 질환을 치료하기 위한 약제의 제조에 있어 상기한 화합물의 용도에 관한 것이다.
The present invention relates to novel carboxylic acid derivatives of 11-oxo-11H-pyrido [2,1-b]quinazoline-6-carboxamide as potent inhibitors of protein kinase, to pharmaceutical compositions containing them and to the use of said compounds for the manufacture of a medicament for the treatment of pathological conditions or diseases which can be improved by the inhibition of protein kinase |
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| AbstractList | 본 발명은 단백질 키나제의 강력한 저해제로서 11-옥소-11H-피리도 [2,1-b]퀴나졸린-6-카르복사미드의 신규한 카르복시산 유도체, 이를 포함하는 약학적 조성물, 및 단백질 키나제를 저해함으로써 개선할 수 있는 질환 또는 병리학적 질환을 치료하기 위한 약제의 제조에 있어 상기한 화합물의 용도에 관한 것이다.
The present invention relates to novel carboxylic acid derivatives of 11-oxo-11H-pyrido [2,1-b]quinazoline-6-carboxamide as potent inhibitors of protein kinase, to pharmaceutical compositions containing them and to the use of said compounds for the manufacture of a medicament for the treatment of pathological conditions or diseases which can be improved by the inhibition of protein kinase |
| Author | KURZ GUIDO CAMACHO GOMEZ JUAN |
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| Snippet | 본 발명은 단백질 키나제의 강력한 저해제로서 11-옥소-11H-피리도 [2,1-b]퀴나졸린-6-카르복사미드의 신규한 카르복시산 유도체, 이를 포함하는 약학적 조성물, 및 단백질 키나제를 저해함으로써 개선할 수 있는 질환 또는 병리학적 질환을 치료하기 위한 약제의 제조에 있어 상기한... |
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| Title | 단백질 키나제 저해제로서 유용한 피리도퀴나졸린의 카르복시산 유도체 |
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