TARP- 8 AMPA 6--3H-13--2- 6-SUBSTITUTED-3H-13-BENZOTHIAZOL-2-ONE COMPOUNDS AS TARP-GAMMA 8 DEPENDENT AMPA RECEPTOR ANTAGONISTS

하기 화학식의 TARP γ8 의존성 AMPA 수용체 길항제; 그의 제약상 허용되는 염, 용도 및 그의 제조 방법이 기재되어 있다.여기서 X는 CH 또는 N이고; A는이고; R은 본원에 정의된 바와 같다. A TARP γ8 dependant AMPA receptor antagonist of the formula: wherein X is CH or N; A is and R1 is as defined herein; its pharmaceutically acceptable salts, uses, and methods for its prep...

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Main Authors SPINAZZE PATRICK GIANPIETRO, REEL JON KEVIN, ORNSTEIN PAUL LESLIE, MAYHUGH DANIEL RAY, PORTER WARREN JAYE, STEVENS FREDDIE CRAIG, WITKIN JEFFREY MICHAEL, HOLLINSHEAD SEAN PATRICK, KHILEVICH ALBERT, SCHKERYANTZ JEFFREY MICHAEL, GERNERT DOUGLAS LINN, HAHN PATRIC JAMES, GARDINIER KEVIN MATTHEW
Format Patent
LanguageEnglish
Korean
Published 09.12.2016
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Abstract 하기 화학식의 TARP γ8 의존성 AMPA 수용체 길항제; 그의 제약상 허용되는 염, 용도 및 그의 제조 방법이 기재되어 있다.여기서 X는 CH 또는 N이고; A는이고; R은 본원에 정의된 바와 같다. A TARP γ8 dependant AMPA receptor antagonist of the formula: wherein X is CH or N; A is and R1 is as defined herein; its pharmaceutically acceptable salts, uses, and methods for its preparation are described.
AbstractList 하기 화학식의 TARP γ8 의존성 AMPA 수용체 길항제; 그의 제약상 허용되는 염, 용도 및 그의 제조 방법이 기재되어 있다.여기서 X는 CH 또는 N이고; A는이고; R은 본원에 정의된 바와 같다. A TARP γ8 dependant AMPA receptor antagonist of the formula: wherein X is CH or N; A is and R1 is as defined herein; its pharmaceutically acceptable salts, uses, and methods for its preparation are described.
Author ORNSTEIN PAUL LESLIE
MAYHUGH DANIEL RAY
STEVENS FREDDIE CRAIG
WITKIN JEFFREY MICHAEL
KHILEVICH ALBERT
SPINAZZE PATRICK GIANPIETRO
GERNERT DOUGLAS LINN
HOLLINSHEAD SEAN PATRICK
REEL JON KEVIN
PORTER WARREN JAYE
HAHN PATRIC JAMES
GARDINIER KEVIN MATTHEW
SCHKERYANTZ JEFFREY MICHAEL
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– fullname: ORNSTEIN PAUL LESLIE
– fullname: MAYHUGH DANIEL RAY
– fullname: PORTER WARREN JAYE
– fullname: STEVENS FREDDIE CRAIG
– fullname: WITKIN JEFFREY MICHAEL
– fullname: HOLLINSHEAD SEAN PATRICK
– fullname: KHILEVICH ALBERT
– fullname: SCHKERYANTZ JEFFREY MICHAEL
– fullname: GERNERT DOUGLAS LINN
– fullname: HAHN PATRIC JAMES
– fullname: GARDINIER KEVIN MATTHEW
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DocumentTitleAlternate TARP-감마 8 의존성 AMPA 수용체 길항제로서의 6-치환된-3H-1,3-벤조티아졸-2-온 화합물
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Snippet 하기 화학식의 TARP γ8 의존성 AMPA 수용체 길항제; 그의 제약상 허용되는 염, 용도 및 그의 제조 방법이 기재되어 있다.여기서 X는 CH 또는 N이고; A는이고; R은 본원에 정의된 바와 같다. A TARP γ8 dependant AMPA receptor antagonist...
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SourceType Open Access Repository
SubjectTerms CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
Title TARP- 8 AMPA 6--3H-13--2- 6-SUBSTITUTED-3H-13-BENZOTHIAZOL-2-ONE COMPOUNDS AS TARP-GAMMA 8 DEPENDENT AMPA RECEPTOR ANTAGONISTS
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