TARP- 8 AMPA 6--3H-13--2- 6-SUBSTITUTED-3H-13-BENZOTHIAZOL-2-ONE COMPOUNDS AS TARP-GAMMA 8 DEPENDENT AMPA RECEPTOR ANTAGONISTS
하기 화학식의 TARP γ8 의존성 AMPA 수용체 길항제; 그의 제약상 허용되는 염, 용도 및 그의 제조 방법이 기재되어 있다.여기서 X는 CH 또는 N이고; A는이고; R은 본원에 정의된 바와 같다. A TARP γ8 dependant AMPA receptor antagonist of the formula: wherein X is CH or N; A is and R1 is as defined herein; its pharmaceutically acceptable salts, uses, and methods for its prep...
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Format | Patent |
Language | English Korean |
Published |
09.12.2016
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Abstract | 하기 화학식의 TARP γ8 의존성 AMPA 수용체 길항제; 그의 제약상 허용되는 염, 용도 및 그의 제조 방법이 기재되어 있다.여기서 X는 CH 또는 N이고; A는이고; R은 본원에 정의된 바와 같다.
A TARP γ8 dependant AMPA receptor antagonist of the formula: wherein X is CH or N; A is and R1 is as defined herein; its pharmaceutically acceptable salts, uses, and methods for its preparation are described. |
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AbstractList | 하기 화학식의 TARP γ8 의존성 AMPA 수용체 길항제; 그의 제약상 허용되는 염, 용도 및 그의 제조 방법이 기재되어 있다.여기서 X는 CH 또는 N이고; A는이고; R은 본원에 정의된 바와 같다.
A TARP γ8 dependant AMPA receptor antagonist of the formula: wherein X is CH or N; A is and R1 is as defined herein; its pharmaceutically acceptable salts, uses, and methods for its preparation are described. |
Author | ORNSTEIN PAUL LESLIE MAYHUGH DANIEL RAY STEVENS FREDDIE CRAIG WITKIN JEFFREY MICHAEL KHILEVICH ALBERT SPINAZZE PATRICK GIANPIETRO GERNERT DOUGLAS LINN HOLLINSHEAD SEAN PATRICK REEL JON KEVIN PORTER WARREN JAYE HAHN PATRIC JAMES GARDINIER KEVIN MATTHEW SCHKERYANTZ JEFFREY MICHAEL |
Author_xml | – fullname: SPINAZZE PATRICK GIANPIETRO – fullname: REEL JON KEVIN – fullname: ORNSTEIN PAUL LESLIE – fullname: MAYHUGH DANIEL RAY – fullname: PORTER WARREN JAYE – fullname: STEVENS FREDDIE CRAIG – fullname: WITKIN JEFFREY MICHAEL – fullname: HOLLINSHEAD SEAN PATRICK – fullname: KHILEVICH ALBERT – fullname: SCHKERYANTZ JEFFREY MICHAEL – fullname: GERNERT DOUGLAS LINN – fullname: HAHN PATRIC JAMES – fullname: GARDINIER KEVIN MATTHEW |
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DocumentTitleAlternate | TARP-감마 8 의존성 AMPA 수용체 길항제로서의 6-치환된-3H-1,3-벤조티아졸-2-온 화합물 |
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Snippet | 하기 화학식의 TARP γ8 의존성 AMPA 수용체 길항제; 그의 제약상 허용되는 염, 용도 및 그의 제조 방법이 기재되어 있다.여기서 X는 CH 또는 N이고; A는이고; R은 본원에 정의된 바와 같다.
A TARP γ8 dependant AMPA receptor antagonist... |
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SubjectTerms | CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES |
Title | TARP- 8 AMPA 6--3H-13--2- 6-SUBSTITUTED-3H-13-BENZOTHIAZOL-2-ONE COMPOUNDS AS TARP-GAMMA 8 DEPENDENT AMPA RECEPTOR ANTAGONISTS |
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