ALPHA-GUANIDINO ACID DERIVATIVE AND ITS PRODUCTION

• Main Authors: UEKI YASUYUKI, KIMURA YUMIKO
• Format: Patent
• Language: English
• Published: 18.01.1994
• Edition: 5
• Subjects: ACYCLIC OR CARBOCYCLIC COMPOUNDS; CHEMISTRY; CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION ORPROCESSING OF GOODS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; METALLURGY; ORGANIC CHEMISTRY; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS; TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINSTCLIMATE CHANGE

PURPOSE:To provide a new alpha-guanidino acid derivative useful for selectively amidinating the N-terminal of a peptide under mild conditions. CONSTITUTION:The compound of formula I [R1 is substituted benzenesulfonyl bearing 1 to 5 methyl or methoxy groups on the benzene ring; R2 is a side chain obt...