PERIPHERAL OPIOID RECEPTOR ANTAGONISTS AND USES THEREOF
To provide peripheral opioid receptor antagonists and formulations containing the same.SOLUTION: The present invention provides a compound represented by formula I in the figure, and formulations containing the same. [In the formula, R1 and R2 are each independently a C1-6 aliphatic group; and X- is...
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Format | Patent |
Language | English Japanese |
Published |
10.12.2020
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Abstract | To provide peripheral opioid receptor antagonists and formulations containing the same.SOLUTION: The present invention provides a compound represented by formula I in the figure, and formulations containing the same. [In the formula, R1 and R2 are each independently a C1-6 aliphatic group; and X- is a suitable anion.]SELECTED DRAWING: None
【課題】末梢オピオイド受容体アンタゴニストおよびそれを含有する製剤の提供。【解決手段】式I:[式中、R1およびR2は、各々独立して、C1−6脂肪族であり;X−は、適当なアニオンである]で示される化合物およびそれを含有する製剤。【選択図】なし |
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AbstractList | To provide peripheral opioid receptor antagonists and formulations containing the same.SOLUTION: The present invention provides a compound represented by formula I in the figure, and formulations containing the same. [In the formula, R1 and R2 are each independently a C1-6 aliphatic group; and X- is a suitable anion.]SELECTED DRAWING: None
【課題】末梢オピオイド受容体アンタゴニストおよびそれを含有する製剤の提供。【解決手段】式I:[式中、R1およびR2は、各々独立して、C1−6脂肪族であり;X−は、適当なアニオンである]で示される化合物およびそれを含有する製剤。【選択図】なし |
Author | GEORGE JOSEPH DONATO III ZHANG HUYI NATALIYA BAZHINA CHRISTIAN OFSLAGER SHAH SYED M JAN SZELIGA JOHN LOKHNAUTH STEVEN R FABIAN NIKETA PATEL GALEN RADEBAUGH TIANMIN ZHU SREENIVASULU MEGATI CHARLES MELUCCI |
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Snippet | To provide peripheral opioid receptor antagonists and formulations containing the same.SOLUTION: The present invention provides a compound represented by... |
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SubjectTerms | CHEMISTRY DEVICES FOR INTRODUCING MEDIA INTO, OR ONTO, THE BODY DEVICES FOR PRODUCING OR ENDING SLEEP OR STUPOR DEVICES FOR TRANSDUCING BODY MEDIA OR FOR TAKING MEDIA FROMTHE BODY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS |
Title | PERIPHERAL OPIOID RECEPTOR ANTAGONISTS AND USES THEREOF |
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