SUSTAINED RELEASE FORMULATION OF A NON-STEROIDAL ANTI-INFLAMMATORY DRUG
PROBLEM TO BE SOLVED: To provide formulations comprising multivesicular liposomes and one or more non-steroidal anti-inflammatory drugs.SOLUTION: Disclosed herein is a formulation comprising multivesicular liposomes and one or more non-steroidal anti-inflammatory drugs, which minimizes the side effe...
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Format | Patent |
Language | English Japanese |
Published |
26.04.2018
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Abstract | PROBLEM TO BE SOLVED: To provide formulations comprising multivesicular liposomes and one or more non-steroidal anti-inflammatory drugs.SOLUTION: Disclosed herein is a formulation comprising multivesicular liposomes and one or more non-steroidal anti-inflammatory drugs, which minimizes the side effects of unencapsulated non-steroidal anti-inflammatory drugs while maintaining or improving efficacy. Methods of making and administering the formulation comprising multivesicular liposomes and one or more non-steroidal anti-inflammatory drugs, and its use as a medicament are also provided.SELECTED DRAWING: None
【課題】多小胞リポソーム、ならびに、1種類あるいはそれよりも多くの種類の、非ステロイド性である抗炎症薬を含む処方物を提供すること【解決手段】多小胞リポソーム、ならびに、1種類あるいはそれよりも多くの種類の、非ステロイド性である抗炎症薬を含む処方物が開示されるものであるところ、ここにおいて、それは、有効性を維持または改善しながら、封入されていない、非ステロイド性である抗炎症薬の副作用を最小限にする。多小胞リポソームおよび1種類あるいはそれよりも多くの種類の、非ステロイド性抗炎症薬を含んでいる処方物を産生および投与する方法、およびその薬物としての使用も提供される。【選択図】なし |
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AbstractList | PROBLEM TO BE SOLVED: To provide formulations comprising multivesicular liposomes and one or more non-steroidal anti-inflammatory drugs.SOLUTION: Disclosed herein is a formulation comprising multivesicular liposomes and one or more non-steroidal anti-inflammatory drugs, which minimizes the side effects of unencapsulated non-steroidal anti-inflammatory drugs while maintaining or improving efficacy. Methods of making and administering the formulation comprising multivesicular liposomes and one or more non-steroidal anti-inflammatory drugs, and its use as a medicament are also provided.SELECTED DRAWING: None
【課題】多小胞リポソーム、ならびに、1種類あるいはそれよりも多くの種類の、非ステロイド性である抗炎症薬を含む処方物を提供すること【解決手段】多小胞リポソーム、ならびに、1種類あるいはそれよりも多くの種類の、非ステロイド性である抗炎症薬を含む処方物が開示されるものであるところ、ここにおいて、それは、有効性を維持または改善しながら、封入されていない、非ステロイド性である抗炎症薬の副作用を最小限にする。多小胞リポソームおよび1種類あるいはそれよりも多くの種類の、非ステロイド性抗炎症薬を含んでいる処方物を産生および投与する方法、およびその薬物としての使用も提供される。【選択図】なし |
Author | WILLIAM JOSEPH LAMBERT GARY PATOU LOUIE DANIEL GARCIA ZHU LIANGJIN |
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DocumentTitleAlternate | 非ステロイド性抗炎症薬の徐放性処方物 |
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Snippet | PROBLEM TO BE SOLVED: To provide formulations comprising multivesicular liposomes and one or more non-steroidal anti-inflammatory drugs.SOLUTION: Disclosed... |
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Title | SUSTAINED RELEASE FORMULATION OF A NON-STEROIDAL ANTI-INFLAMMATORY DRUG |
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