Biarylmethyl heterocycles
The present invention provides compounds of Formula (I):wherein all variables are as defined in the specification, and compositions comprising any of such novel compounds. These compounds are biased agonists, or β-Arrestin agonists of the angiotensin II receptor, which may be used as medicaments.
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| Main Authors | , , , , , , , , , , |
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| Format | Patent |
| Language | English Hebrew |
| Published |
31.01.2019
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| Online Access | Get full text |
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| Abstract | The present invention provides compounds of Formula (I):wherein all variables are as defined in the specification, and compositions comprising any of such novel compounds. These compounds are biased agonists, or β-Arrestin agonists of the angiotensin II receptor, which may be used as medicaments. |
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| AbstractList | The present invention provides compounds of Formula (I):wherein all variables are as defined in the specification, and compositions comprising any of such novel compounds. These compounds are biased agonists, or β-Arrestin agonists of the angiotensin II receptor, which may be used as medicaments. |
| Author | HALPERN Oz Scott TRIPATHY Sasmita PRIESTLEY Eldon Scott RICHTER Jeremy ZHANG Xiaojun RUEL Rejean REZNIK Samuel Kaye RUEDIGER Edward H YANG Wu JIANG Wen GILLARD James R |
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| RelatedCompanies | HALPERN Oz Scott RICHTER Jeremy ZHANG Xiaojun REZNIK Samuel Kaye RUEDIGER Edward H GILLARD James R TRIPATHY Sasmita PRIESTLEY Eldon Scott RUEL Rejean BRISTOL-MYERS SQUIBB COMPANY UNIVERSITE DE MONTREAL YANG Wu JIANG Wen |
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| Snippet | The present invention provides compounds of Formula (I):wherein all variables are as defined in the specification, and compositions comprising any of such... |
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| Title | Biarylmethyl heterocycles |
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