NUEVOS DERIVADOS DE 8HETEROCICLO-PIPERIDINA CONDENSADA)-( PIPERAZINIL)-1-ALCANONA O DE (HETEROCICLO-PIRROLIDINA CONDENSADA)-(PIPERAZINIL)-1-ALCANONA Y SU UTILIZACION COMO INHIBIDORES DE P75
LA INVENCION SE REFIERE A DERIVADOS DE (HETEROCICLO-PIPERIDINA CONDENSADAS)-(PIPERAZINIL)-1-ALCANONA Y A (HETEROCICLO-PIRROLIDINA CONDENSADAS)-(PIPERAZINIL)-1-ALCANONA DE FORMULA GENERAL (1) EN LA QUE A,W,N Y R2 SON TALES COMO SE DEFINEN EN LA REIVINDICACION 1, ASI COMO SU PROCEDIMIENTO DE PREPARACI...
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Format | Patent |
Language | Spanish |
Published |
13.07.2015
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Abstract | LA INVENCION SE REFIERE A DERIVADOS DE (HETEROCICLO-PIPERIDINA CONDENSADAS)-(PIPERAZINIL)-1-ALCANONA Y A (HETEROCICLO-PIRROLIDINA CONDENSADAS)-(PIPERAZINIL)-1-ALCANONA DE FORMULA GENERAL (1) EN LA QUE A,W,N Y R2 SON TALES COMO SE DEFINEN EN LA REIVINDICACION 1, ASI COMO SU PROCEDIMIENTO DE PREPARACION Y SU APLICACION EN TERAPEUTICA.
The disclosure relates to (heterocycle-fused piperidine)-(piperazinyl)-1-alkanone derivatives and (heterocycle-fused pyrrolidine)-(piperazinyl)-1-alkanone derivatives of formula (I): wherein A, W, R2 and n are as defined in the disclosure, to the method of preparation thereof and the therapeutic use thereof. |
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AbstractList | LA INVENCION SE REFIERE A DERIVADOS DE (HETEROCICLO-PIPERIDINA CONDENSADAS)-(PIPERAZINIL)-1-ALCANONA Y A (HETEROCICLO-PIRROLIDINA CONDENSADAS)-(PIPERAZINIL)-1-ALCANONA DE FORMULA GENERAL (1) EN LA QUE A,W,N Y R2 SON TALES COMO SE DEFINEN EN LA REIVINDICACION 1, ASI COMO SU PROCEDIMIENTO DE PREPARACION Y SU APLICACION EN TERAPEUTICA.
The disclosure relates to (heterocycle-fused piperidine)-(piperazinyl)-1-alkanone derivatives and (heterocycle-fused pyrrolidine)-(piperazinyl)-1-alkanone derivatives of formula (I): wherein A, W, R2 and n are as defined in the disclosure, to the method of preparation thereof and the therapeutic use thereof. |
Author | MARCO BARONI FRANCOISE BONO SANDRINE DELBARY-GOSSART VALENTINA VERCESI |
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Snippet | LA INVENCION SE REFIERE A DERIVADOS DE (HETEROCICLO-PIPERIDINA CONDENSADAS)-(PIPERAZINIL)-1-ALCANONA Y A (HETEROCICLO-PIRROLIDINA... |
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Title | NUEVOS DERIVADOS DE 8HETEROCICLO-PIPERIDINA CONDENSADA)-( PIPERAZINIL)-1-ALCANONA O DE (HETEROCICLO-PIRROLIDINA CONDENSADA)-(PIPERAZINIL)-1-ALCANONA Y SU UTILIZACION COMO INHIBIDORES DE P75 |
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