DERIVADOS DE 4-ARILMORFOLIN-3-ONA, SU PREPARACION Y SU APLICACION EN TERAPEUTICA
LA PRESENTE INVENCION TIENE POR OBJETO NUEVOS DERIVADOS DE 4-ARILMORFOLIN-3-ONA, SU PREPARACION Y SU APLICACION EN TERAPOUTICA.- LOS COMPUESTOS PRESENTAN UNA IMPORTANTE AFINIDAD CON LOS RECEPTORES "NK2" HUMANOS DE LA NEUROQUININA A.- LA NEUROQUININA "A (NKA) PERTENE AL GRUPO DE NEUROP...
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Format | Patent |
Language | Spanish |
Published |
14.05.2009
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Online Access | Get full text |
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Abstract | LA PRESENTE INVENCION TIENE POR OBJETO NUEVOS DERIVADOS DE 4-ARILMORFOLIN-3-ONA, SU PREPARACION Y SU APLICACION EN TERAPOUTICA.- LOS COMPUESTOS PRESENTAN UNA IMPORTANTE AFINIDAD CON LOS RECEPTORES "NK2" HUMANOS DE LA NEUROQUININA A.- LA NEUROQUININA "A (NKA) PERTENE AL GRUPO DE NEUROPOPTIDOS LLAMADOS TAQUIQUININAS O NEUROQUININAS QUE INCLUYE LA SUBSTANCIA "p" (SP) Y LA NEUROQUININA B (NKB).- LA PRESENTE INVENCION TIENE POR OBJETO LOS COMPUESTOS UE RESPONDEN A LA FORMULA I (Vease formula)
The invention relates to compounds corresponding to formula (I): in which: Ar represents a mono- or disubstituted phenyl; R1 represents an unsubstituted or substituted phenyl; R2 represents: a pyridyl; an unsubstituted or substituted phenyl; a benzyl that is unsubstituted or substituted on the phenyl; R2 may moreover represent: a heterocyclic radical; R3 represents various values. The invention also comprises methods for the compounds preparation, formulations comprising them and therapeutic applications thereof. |
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AbstractList | LA PRESENTE INVENCION TIENE POR OBJETO NUEVOS DERIVADOS DE 4-ARILMORFOLIN-3-ONA, SU PREPARACION Y SU APLICACION EN TERAPOUTICA.- LOS COMPUESTOS PRESENTAN UNA IMPORTANTE AFINIDAD CON LOS RECEPTORES "NK2" HUMANOS DE LA NEUROQUININA A.- LA NEUROQUININA "A (NKA) PERTENE AL GRUPO DE NEUROPOPTIDOS LLAMADOS TAQUIQUININAS O NEUROQUININAS QUE INCLUYE LA SUBSTANCIA "p" (SP) Y LA NEUROQUININA B (NKB).- LA PRESENTE INVENCION TIENE POR OBJETO LOS COMPUESTOS UE RESPONDEN A LA FORMULA I (Vease formula)
The invention relates to compounds corresponding to formula (I): in which: Ar represents a mono- or disubstituted phenyl; R1 represents an unsubstituted or substituted phenyl; R2 represents: a pyridyl; an unsubstituted or substituted phenyl; a benzyl that is unsubstituted or substituted on the phenyl; R2 may moreover represent: a heterocyclic radical; R3 represents various values. The invention also comprises methods for the compounds preparation, formulations comprising them and therapeutic applications thereof. |
Author | XAVIER EMONDS-ALT VINCENZO PROIETTO |
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Snippet | LA PRESENTE INVENCION TIENE POR OBJETO NUEVOS DERIVADOS DE 4-ARILMORFOLIN-3-ONA, SU PREPARACION Y SU APLICACION EN TERAPOUTICA.- LOS COMPUESTOS PRESENTAN UNA... |
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Title | DERIVADOS DE 4-ARILMORFOLIN-3-ONA, SU PREPARACION Y SU APLICACION EN TERAPEUTICA |
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