PYRAZOLO[1,5-A]PYRAZINE DERIVATIVES AS BTK INHIBITORS

Provided are compounds of Formula (I'): or pharmaceutically acceptable salts thereof, wherein the variables in the formula are as defined herein; and methods for their use and production.

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Main Authors PRINCE, Robin, MARX, Isaac, LIN, Edward, Yin-shiang, PATTAROPONG, Vatee, CAPACCI, Andrew, George, JONES, John, Howard, SCHULZ, Jurgen, VANDEVEER, George, YOUSAF, Zain, HIMMELBAUER, Martin, HOPKINS, Brian, T, CHEN, Teyu, MA, Bin, NEVALAINEN, Marta, GONZALEZ LOPEZ DE TURISO, Felix, PURGETT, Thomas, SCIABOLA, Simone
Format Patent
LanguageEnglish
French
German
Published 20.09.2023
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Abstract Provided are compounds of Formula (I'): or pharmaceutically acceptable salts thereof, wherein the variables in the formula are as defined herein; and methods for their use and production.
AbstractList Provided are compounds of Formula (I'): or pharmaceutically acceptable salts thereof, wherein the variables in the formula are as defined herein; and methods for their use and production.
Author PURGETT, Thomas
MARX, Isaac
CHEN, Teyu
PRINCE, Robin
NEVALAINEN, Marta
PATTAROPONG, Vatee
HIMMELBAUER, Martin
HOPKINS, Brian, T
JONES, John, Howard
VANDEVEER, George
SCIABOLA, Simone
YOUSAF, Zain
SCHULZ, Jurgen
LIN, Edward, Yin-shiang
MA, Bin
CAPACCI, Andrew, George
GONZALEZ LOPEZ DE TURISO, Felix
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– fullname: LIN, Edward, Yin-shiang
– fullname: PATTAROPONG, Vatee
– fullname: CAPACCI, Andrew, George
– fullname: JONES, John, Howard
– fullname: SCHULZ, Jurgen
– fullname: VANDEVEER, George
– fullname: YOUSAF, Zain
– fullname: HIMMELBAUER, Martin
– fullname: HOPKINS, Brian, T
– fullname: CHEN, Teyu
– fullname: MA, Bin
– fullname: NEVALAINEN, Marta
– fullname: GONZALEZ LOPEZ DE TURISO, Felix
– fullname: PURGETT, Thomas
– fullname: SCIABOLA, Simone
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DocumentTitleAlternate PYRAZOLO[1,5-A PYRAZINDERIVATE ALS BTK INHIBITOREN
DÉRIVÉS DE PYRAZOLO[1,5-A]PYRAZINE UTILISÉS EN TANT QU'INHIBITEURS DE BTK
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Snippet Provided are compounds of Formula (I'): or pharmaceutically acceptable salts thereof, wherein the variables in the formula are as defined herein; and methods...
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SubjectTerms CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
Title PYRAZOLO[1,5-A]PYRAZINE DERIVATIVES AS BTK INHIBITORS
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