MODULATORS OF THE BETA-3 ADRENERGIC RECEPTOR USEFUL FOR THE TREATMENT OR PREVENTION OF HEART FAILURE AND DISORDERS RELATED THERETO
The present invention relates to compounds of Formula (Ia) and pharmaceutical compositions thereof that modulate the activity of the beta-3 adrenergic receptor. Compounds of the present invention and pharmaceutical compositions thereof are directed to methods useful in the treatment of a beta-3 adre...
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| Main Authors | , , , , |
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| Format | Patent |
| Language | English French German |
| Published |
14.10.2020
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| Online Access | Get full text |
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| Abstract | The present invention relates to compounds of Formula (Ia) and pharmaceutical compositions thereof that modulate the activity of the beta-3 adrenergic receptor. Compounds of the present invention and pharmaceutical compositions thereof are directed to methods useful in the treatment of a beta-3 adrenergic receptor-mediated disorder, such as, heart failure and related disorders thereto. |
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| AbstractList | The present invention relates to compounds of Formula (Ia) and pharmaceutical compositions thereof that modulate the activity of the beta-3 adrenergic receptor. Compounds of the present invention and pharmaceutical compositions thereof are directed to methods useful in the treatment of a beta-3 adrenergic receptor-mediated disorder, such as, heart failure and related disorders thereto. |
| Author | TRAN, Thuy-Anh KRAMER, Bryan Aubrey ULLMAN, Brett SHIN, Young-Jun DO, Quyen-Quyen Thuy |
| Author_xml | – fullname: ULLMAN, Brett – fullname: TRAN, Thuy-Anh – fullname: DO, Quyen-Quyen Thuy – fullname: KRAMER, Bryan Aubrey – fullname: SHIN, Young-Jun |
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| DocumentTitleAlternate | MODULATOREN DES BETA-3-ADRENERGEN REZEPTORS NÜTZLICH ZUR BEHANDLUNG ODER PRÄVENTION VON HERZINSUFFIZIENZ UND DAMIT ASSOZIIERTEN ERKRANKUNGEN MODULATEURS DU RÉCEPTEUR ADRÉNERGIQUE BÊTA 3 UTILE DANS LE TRAITEMENT OU LA PRÉVENTION DE L'INSUFFISANCE CARDIAQUE ET DE TROUBLES ASSOCIÉS À CELLE-CI |
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| PublicationYear | 2020 |
| RelatedCompanies | Arena Pharmaceuticals, Inc |
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| Snippet | The present invention relates to compounds of Formula (Ia) and pharmaceutical compositions thereof that modulate the activity of the beta-3 adrenergic... |
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| Title | MODULATORS OF THE BETA-3 ADRENERGIC RECEPTOR USEFUL FOR THE TREATMENT OR PREVENTION OF HEART FAILURE AND DISORDERS RELATED THERETO |
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