PROCESS AND INTERMEDIATES FOR PREPARING PRODRUGS OF PYRIDONE AMIDES USEFUL AS MODULATORS OF SODIUM CHANNELS

The invention relates to a process and intermediates for preparing prodrug compounds of formula I: wherein R2, R3, R5, R7 and X are as defined herein.

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Bibliographic Details
Main Authors ANDERSON, Corey, HADIDA-RUAH, Sara Sabina, LITTLER, Benjamin Joseph, KESHAVARZ-SHOKRI, Ali, ALCACIO, Tim Edward, ZHANG, Beili, GOLEC, Julian Marian Charles, BELMONT, Daniel T
Format Patent
LanguageEnglish
French
German
Published 07.08.2024
Subjects
ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAININGELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN,SULFUR, SELENIUM OR TELLURIUM
CHEMISTRY
METALLURGY
ORGANIC CHEMISTRY
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Abstract The invention relates to a process and intermediates for preparing prodrug compounds of formula I: wherein R2, R3, R5, R7 and X are as defined herein.
AbstractList The invention relates to a process and intermediates for preparing prodrug compounds of formula I: wherein R2, R3, R5, R7 and X are as defined herein.
Author GOLEC, Julian Marian Charles
LITTLER, Benjamin Joseph
ALCACIO, Tim Edward
HADIDA-RUAH, Sara Sabina
ZHANG, Beili
KESHAVARZ-SHOKRI, Ali
ANDERSON, Corey
BELMONT, Daniel T
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– fullname: HADIDA-RUAH, Sara Sabina
– fullname: LITTLER, Benjamin Joseph
– fullname: KESHAVARZ-SHOKRI, Ali
– fullname: ALCACIO, Tim Edward
– fullname: ZHANG, Beili
– fullname: GOLEC, Julian Marian Charles
– fullname: BELMONT, Daniel T
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DocumentTitleAlternate PROCÉDÉ ET INTERMÉDIAIRES POUR LA PRÉPARATION DES PROMÉDICAMENTS D'AMIDES DE PYRIDONE UTILES EN TANT QUE MODULATEURS DE CANAUX SODIQUES
PROZESS UND INTERMEDIATE ZUR HERSTELLUNG VON PRODRUGS VON PYRIDONAMIDEN ALS NATRIUMKANALMODULATOREN
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RelatedCompanies Vertex Pharmaceuticals Incorporated
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Snippet The invention relates to a process and intermediates for preparing prodrug compounds of formula I: wherein R2, R3, R5, R7 and X are as defined herein.
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SubjectTerms ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAININGELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN,SULFUR, SELENIUM OR TELLURIUM
CHEMISTRY
METALLURGY
ORGANIC CHEMISTRY
Title PROCESS AND INTERMEDIATES FOR PREPARING PRODRUGS OF PYRIDONE AMIDES USEFUL AS MODULATORS OF SODIUM CHANNELS
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