5-ARYL-1-IMINO-1-OXO-[1,2,4]THIADIAZINES
The present invention provides a compound of formula I' having BACE1 inhibitory activity, their manufacture, pharmaceutical compositions containing them and their use as therapeutically active substances. The active compounds of the present invention are useful in the therapeutic and/or prophyl...
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| Main Authors | , , , , , , , |
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| Format | Patent |
| Language | English French German |
| Published |
13.03.2019
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| Subjects | |
| Online Access | Get full text |
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| Abstract | The present invention provides a compound of formula I' having BACE1 inhibitory activity, their manufacture, pharmaceutical compositions containing them and their use as therapeutically active substances. The active compounds of the present invention are useful in the therapeutic and/or prophylactic treatment of e.g. Alzheimer's disease. |
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| AbstractList | The present invention provides a compound of formula I' having BACE1 inhibitory activity, their manufacture, pharmaceutical compositions containing them and their use as therapeutically active substances. The active compounds of the present invention are useful in the therapeutic and/or prophylactic treatment of e.g. Alzheimer's disease. |
| Author | WERMUTH, Roger SCHNIDER, Christian GUBA, Wolfgang PETERS, Jens-Uwe OBST SANDER, Ulrike HAAP, Wolfgang KUGLSTATTER, Andreas WOLTERING, Thomas |
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| RelatedCompanies | F. Hoffmann-La Roche AG |
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| Snippet | The present invention provides a compound of formula I' having BACE1 inhibitory activity, their manufacture, pharmaceutical compositions containing them and... |
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| Title | 5-ARYL-1-IMINO-1-OXO-[1,2,4]THIADIAZINES |
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