SUBSTITUTED ARYLSULPHONYLGLYCINES, THE PREPARATION THEREOF AND THE USE THEREOF AS PHARMACEUTICAL COMPOSITIONS
The present invention relates to substituted arylsulphonylglycines of general formula wherein R, R4, X, Y, Z and m are defined as in claim 1, the tautomers, enantiomers, diastereomers, mixtures thereof and salts thereof, which have valuable pharmacological properties, particularly the suppression of...
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Format | Patent |
Language | English French German |
Published |
18.07.2012
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Abstract | The present invention relates to substituted arylsulphonylglycines of general formula wherein R, R4, X, Y, Z and m are defined as in claim 1, the tautomers, enantiomers, diastereomers, mixtures thereof and salts thereof, which have valuable pharmacological properties, particularly the suppression of the interaction of glycogen phosphorylase a with the GL subunit of glycogen-associated protein phosphatase 1 (PP1), and their use as pharmaceutical compositions. |
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AbstractList | The present invention relates to substituted arylsulphonylglycines of general formula wherein R, R4, X, Y, Z and m are defined as in claim 1, the tautomers, enantiomers, diastereomers, mixtures thereof and salts thereof, which have valuable pharmacological properties, particularly the suppression of the interaction of glycogen phosphorylase a with the GL subunit of glycogen-associated protein phosphatase 1 (PP1), and their use as pharmaceutical compositions. |
Author | SCHOELCH, CORINNA WAGNER, HOLGER STREICHER, RUEDIGER SCHULER-METZ, ANNETTE ECKHARDT, MATTHIAS LANGKOPF, ELKE PAUTSCH, ALEXANDER |
Author_xml | – fullname: SCHOELCH, CORINNA – fullname: WAGNER, HOLGER – fullname: ECKHARDT, MATTHIAS – fullname: PAUTSCH, ALEXANDER – fullname: SCHULER-METZ, ANNETTE – fullname: LANGKOPF, ELKE – fullname: STREICHER, RUEDIGER |
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DocumentTitleAlternate | NOUVELLES ARYLSULPHONYLGLYCINES SUBSTITUÉES, LEUR PROCÉDÉ DE PRÉPARATION ET LEUR UTILISATION EN TANT QUE COMPOSITIONS PHARMACEUTIQUES SUBSTITUIERTE ARYLSULPHONYLGLYCINE, IHRE HERSTELLUNG UND IHRE VERWENDUNG ALS PHARMAZEUTISCHE ZUSAMMENSETZUNGEN |
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Snippet | The present invention relates to substituted arylsulphonylglycines of general formula wherein R, R4, X, Y, Z and m are defined as in claim 1, the tautomers,... |
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Title | SUBSTITUTED ARYLSULPHONYLGLYCINES, THE PREPARATION THEREOF AND THE USE THEREOF AS PHARMACEUTICAL COMPOSITIONS |
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