PIPERIDINES AND PYRROLIDINES

The invention relates to novel piperidine and pyrrolidine derivatives of formula (I) in which R , R , R , k, l, m and n have the meanings indicated in Claim 1, and their salts, novel intermediates and processes for the preparation of the compounds according to the invention. The compounds of formula...

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Main Authors GREINER HARTMUT, BOTTCHER HENNING, HARTING JURGEN, MARZ JOACHIM, HANSSON LARS OLOV, SEYFRIED CHRISTOPH, SONESSON CLAS AKE, DEVANT RALF, BARTOSZYK GERD, BENGT RONNY ANDERSSON, STJERNLOF NILS PETER
Format Patent
LanguageCzech
English
Published 13.01.1999
Edition6
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Abstract The invention relates to novel piperidine and pyrrolidine derivatives of formula (I) in which R , R , R , k, l, m and n have the meanings indicated in Claim 1, and their salts, novel intermediates and processes for the preparation of the compounds according to the invention. The compounds of formula (I) act as 5-HT1A receptor antagonists and exhibit 5-HT reuptake-inhibiting actions and can be used for the production of medicaments.
AbstractList The invention relates to novel piperidine and pyrrolidine derivatives of formula (I) in which R , R , R , k, l, m and n have the meanings indicated in Claim 1, and their salts, novel intermediates and processes for the preparation of the compounds according to the invention. The compounds of formula (I) act as 5-HT1A receptor antagonists and exhibit 5-HT reuptake-inhibiting actions and can be used for the production of medicaments.
Author HANSSON LARS OLOV
GREINER HARTMUT
BOTTCHER HENNING
SONESSON CLAS AKE
HARTING JURGEN
SEYFRIED CHRISTOPH
MARZ JOACHIM
BARTOSZYK GERD
DEVANT RALF
STJERNLOF NILS PETER
BENGT RONNY ANDERSSON
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– fullname: SEYFRIED CHRISTOPH
– fullname: SONESSON CLAS AKE
– fullname: DEVANT RALF
– fullname: BARTOSZYK GERD
– fullname: BENGT RONNY ANDERSSON
– fullname: STJERNLOF NILS PETER
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DocumentTitleAlternate Piperidiny a pyrrolidiny
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Snippet The invention relates to novel piperidine and pyrrolidine derivatives of formula (I) in which R , R , R , k, l, m and n have the meanings indicated in Claim 1,...
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SubjectTerms CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
Title PIPERIDINES AND PYRROLIDINES
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