METHOD OF PRODUCING NOVEL 2-AMINOCARBONYL-6-ARYL-4H-S-TRIAZOLE1,5-A/ /1,4/BENZDIAZEPINES

Title cpds. are of formula (I): where Q = CONR2R3; R' = H or 1-3C alkyl; R2 and R3 = H, 1-6C alkyl, 2-6C hydroxyalkyl, 4-7C dialkylamino-alkyl, or 7-9C aralkyl, or NR2R3 forms a is not >10C cyclic residue opt. contng. O or NR, where R = 1-4C alkyl or hydroxyalkyl; and rings A and B are opt s...

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Bibliographic Details
Main Authors HECKENDORN,ROLAND,CH, CAGNEUX,ANDRE,CH, MEIER,RENE,CH
Format Patent
LanguageEnglish
Published 29.12.1978
Edition2
Subjects
ADHESIVES
CHEMISTRY
DYES
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
LAKES
MEDICAL OR VETERINARY SCIENCE
METALLURGY
MISCELLANEOUS APPLICATIONS OF MATERIALS
MISCELLANEOUS COMPOSITIONS
MORDANTS
NATURAL RESINS
ORGANIC CHEMISTRY
ORGANIC DYES OR CLOSELY-RELATED COMPOUNDS FOR PRODUCING DYES
PAINTS
POLISHES
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
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Summary:Title cpds. are of formula (I): where Q = CONR2R3; R' = H or 1-3C alkyl; R2 and R3 = H, 1-6C alkyl, 2-6C hydroxyalkyl, 4-7C dialkylamino-alkyl, or 7-9C aralkyl, or NR2R3 forms a is not >10C cyclic residue opt. contng. O or NR, where R = 1-4C alkyl or hydroxyalkyl; and rings A and B are opt subst. by F, Cl, Br, 1-6C alkyl, 1-6C alkoxy, CF3 or NO2; and include salts and 5-N-oxides of I. I are prepd. (a) by condensing HNR3R2 with a deriv. of I (Q = CO2H) or (reductively) with I (Q = CHO), or (b) by cyclizing a 2-(1H-1,2,4-1-rinzolo-3-carboxylic amide-5-halomethyl) substd. benzophenone, or other suitable deriv.
Bibliography:Application Number: CS19760006547