SYNTHETIC PROCESS AND NOVEL INTERMEDIATES

The present disclosure describes a synthetic process and novel intermediates related to spirocyclic azetidenyl-isobenzofuran derivatives having an isothiazoline moiety, which are useful as antiparasitics. La présente invention concerne un procédé de synthèse et de nouveaux intermédiaires associés à...

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Main Authors PERALES, JOE B, PANDI, BHARATHI, BECK, BRENT CHRISTOPHER, SPEAKE, JASON D
Format Patent
LanguageEnglish
French
Published 06.08.2020
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Abstract The present disclosure describes a synthetic process and novel intermediates related to spirocyclic azetidenyl-isobenzofuran derivatives having an isothiazoline moiety, which are useful as antiparasitics. La présente invention concerne un procédé de synthèse et de nouveaux intermédiaires associés à des dérivés d'azétidényl-isobenzofurane spirocycliques ayant une fraction d'isothiazoline, qui sont utiles en tant qu'antiparasitaires.
AbstractList The present disclosure describes a synthetic process and novel intermediates related to spirocyclic azetidenyl-isobenzofuran derivatives having an isothiazoline moiety, which are useful as antiparasitics. La présente invention concerne un procédé de synthèse et de nouveaux intermédiaires associés à des dérivés d'azétidényl-isobenzofurane spirocycliques ayant une fraction d'isothiazoline, qui sont utiles en tant qu'antiparasitaires.
Author PERALES, JOE B
SPEAKE, JASON D
BECK, BRENT CHRISTOPHER
PANDI, BHARATHI
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Snippet The present disclosure describes a synthetic process and novel intermediates related to spirocyclic azetidenyl-isobenzofuran derivatives having an...
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CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
Title SYNTHETIC PROCESS AND NOVEL INTERMEDIATES
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