FSH RECEPTOR ANTAGONISTS
The invention relates to FSH receptor antagonist according to general formula I or a pharmaceutically acceptable salt thereof and to a pharmaceutical composition containing the same. The compounds can be used for the treatment and prevention of endometriosis, for the treatment and prevention of pre-...
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| Main Authors | , , , , , , |
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| Format | Patent |
| Language | English French |
| Published |
19.03.2019
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| Subjects | |
| Online Access | Get full text |
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| Abstract | The invention relates to FSH receptor antagonist according to general formula I or a pharmaceutically acceptable salt thereof and to a pharmaceutical composition containing the same. The compounds can be used for the treatment and prevention of endometriosis, for the treatment and prevention of pre-menopausal and peri-menopausal hormone-dependent breast cancer, for contraception, and for the treatment of uterine fibroids and other menstrual-related disorders.
L'invention concerne un antagoniste du récepteur de la FSH de formule générale (I) ou un sel pharmaceutiquement acceptable de celui-ci, ainsi qu'une composition pharmaceutique le contenant. Ces composés peuvent être utilisés pour le traitement et la prévention de l'endométriose, pour le traitement et la prévention du cancer du sein hormono-dépendant pré-ménopausique et péri-ménopausique, pour la contraception et pour le traitement de fibromes utérins et d'autres troubles liés au cycle menstruel. |
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| AbstractList | The invention relates to FSH receptor antagonist according to general formula I or a pharmaceutically acceptable salt thereof and to a pharmaceutical composition containing the same. The compounds can be used for the treatment and prevention of endometriosis, for the treatment and prevention of pre-menopausal and peri-menopausal hormone-dependent breast cancer, for contraception, and for the treatment of uterine fibroids and other menstrual-related disorders.
L'invention concerne un antagoniste du récepteur de la FSH de formule générale (I) ou un sel pharmaceutiquement acceptable de celui-ci, ainsi qu'une composition pharmaceutique le contenant. Ces composés peuvent être utilisés pour le traitement et la prévention de l'endométriose, pour le traitement et la prévention du cancer du sein hormono-dépendant pré-ménopausique et péri-ménopausique, pour la contraception et pour le traitement de fibromes utérins et d'autres troubles liés au cycle menstruel. |
| Author | BLACKABY, WESLEY PETER ENTHOVEN, MARK HINCHLIFFE, PAUL STUART DEKORT, MARTIN TIMMERS, CORNELIS MARIUS POULIE, CHRISTIAN BERNARD MATTHIJS VERKAIK, SASKIA |
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| DocumentTitleAlternate | ANTAGONISTES DU RECEPTEUR DE LA FSH |
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| RelatedCompanies | MERCK SHARP & DOHME B.V |
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| Snippet | The invention relates to FSH receptor antagonist according to general formula I or a pharmaceutically acceptable salt thereof and to a pharmaceutical... |
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| Title | FSH RECEPTOR ANTAGONISTS |
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